SCHEMBL9056669

SCHEMBL9056669

CCOCCn1cc(C(=O)N2CCC(n3c(C)nc4cnccc43)CC2C)c2c(Cl)cccc21

nearest known ligand 0.74

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
CCR5 P51681 2/20 0.38
CYP2D6 P10635 1/20 0.38
CYP3A4 P08684 2/20 0.36
P2RX7 Q99572 6/20 0.35
IL1B P01584 2/20 0.35
HSD11B1 P28845 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7834134 0.85 CCR5 (0.45) CCR5CYP2D6CYP3A4P2RX7IL1B
SCHEMBL7844030 0.80 P2RX7 (0.38) CYP3A4P2RX7IL1B
Hydrochloric Acid SCHEMBL7847822 0.79 P2RX7 (0.38) CYP3A4P2RX7IL1B
SCHEMBL7835611 0.78 CCR5 (0.46) CCR5CYP2D6CYP3A4
SCHEMBL7835350 0.76 CYP2D6 (0.44) CCR5CYP2D6
SCHEMBL7845819 0.74 CCR5 (0.44) CCR5CYP2D6CYP3A4
SCHEMBL7497419 0.74
SCHEMBL7834484 0.69
SCHEMBL4134368 0.66 CCR5 (0.54) CCR5CYP2D6
SCHEMBL7844278 0.65 CCR5 (0.48) CCR5CYP2D6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1996033196-A1 INDOLE-3-CARBONYL AND INDOLE-3-SULFONYL DERIVATIVES AS PLATELET ACTIVATING FACTOR ANTAGONISTS ABBOTT LABORATORIES (US) 1996-10-24 WO claimed