SCHEMBL7845853

SCHEMBL7845853

c1cnc(-c2cc3ncccc3s2)nc1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP19A1 P11511 3/20 0.44
ALOX5 P09917 1/20 0.40
KDM4E B2RXH2 6/20 0.38
NPC1 O15118 5/20 0.38
RAB9A P51151 5/20 0.38
ALDH1A1 P00352 4/20 0.38
TP53 P04637 1/20 0.38
TSHR P16473 1/20 0.38
SMN1; SMN2 Q16637 1/20 0.38
HSD17B10 Q99714 1/20 0.38
MAPT P10636 2/20 0.38
GLA P06280 1/20 0.38
PIK3CD O00329 1/20 0.38
PIP5K1C O60331 1/20 0.38
PI4KA P42356 1/20 0.38
PIK3CG P48736 1/20 0.38
PI4KB Q9UBF8 1/20 0.38
GRIN3B O60391 1/20 0.38
GRIN1 Q05586 1/20 0.38
GRIN2C Q14957 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL31324900 1.00 CYP19A1 (0.44) CYP19A1ALOX5KDM4ENPC1RAB9A
SCHEMBL28017683 0.90 ALOX5 (0.43) CYP19A1ALOX5KDM4ENPC1RAB9A
SCHEMBL31324889 0.81 NPC1 (0.47) CYP19A1ALOX5KDM4ENPC1RAB9A
SCHEMBL4824051 0.81 IKBKB (0.46) KDM4ENPC1RAB9AALDH1A1TP53
SCHEMBL29987215 0.79 IKBKB (0.45) KDM4ENPC1RAB9AALDH1A1TP53
SCHEMBL3753723 0.77 RAB9A (0.60) CYP19A1KDM4ENPC1RAB9AALDH1A1
SCHEMBL27852488 0.77 ALOX5 (0.36) CYP19A1ALOX5KDM4ENPC1RAB9A
SCHEMBL29022729 0.77 NPC1 (0.46) ALOX5KDM4ENPC1RAB9AALDH1A1
SCHEMBL25165715 0.76 CYP19A1 (0.39) CYP19A1KDM4ENPC1RAB9AALDH1A1
SCHEMBL2581028 0.76 CYP19A1 (0.64) CYP19A1PIK3CDPIK3CG

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1136493-A1 2-(Thienopyridinyl)pyrimidone, 2-(furopyridinyl)pyrimidone 2-(isoquinolinyl)pyrimidone, 2-(pyridoindolyl)pyrimidone and 2-(benzofuropyridinyl)pyrimidone derivatives SANOFI-SYNTHELABO (FR) 2001-09-26 EP disclosed