SCHEMBL7845874

SCHEMBL7845874

CCCCc1cc(N)n2nc(C)cc2n1

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 6/20 0.51
NOS2 P35228 2/20 0.47
TLR7 Q9NYK1 3/20 0.42
ALDH1A1 P00352 6/20 0.42
HPGD P15428 5/20 0.42
NPC1 O15118 4/20 0.42
RAB9A P51151 4/20 0.42
SMN1; SMN2 Q16637 4/20 0.42
NFKB1 P19838 1/20 0.42
HTT P42858 1/20 0.42
NFKB2 Q00653 1/20 0.42
RELA Q04206 1/20 0.42
MAPT P10636 3/20 0.40
MEN1 O00255 2/20 0.40
KMT2A Q03164 2/20 0.40
LMNA P02545 2/20 0.40
TP53 P04637 1/20 0.40
CYP2C19 P33261 1/20 0.40
NPSR1 Q6W5P4 1/20 0.39
PKM P14618 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7847399 0.88 TLR7 (0.48) KDM4ENOS2TLR7ALDH1A1HPGD
SCHEMBL8568147 0.82 NOS2 (0.41) KDM4ENOS2TLR7NPC1RAB9A
SCHEMBL7842532 0.80 NPC1 (0.62) KDM4ETLR7ALDH1A1HPGDNPC1
SCHEMBL7845174 0.76 CDK7 (0.54) NOS2TLR7HRH2HRH3CCNT1
SCHEMBL14088335 0.75 KDM4E (0.43) KDM4ETLR7HPGDNPC1RAB9A
SCHEMBL10623184 0.75 KDM4E (0.43) KDM4ETLR7HPGDNPC1RAB9A
SCHEMBL14099740 0.75 KDM4E (0.43) KDM4ETLR7HPGDNPC1RAB9A
SCHEMBL14182277 0.75 KDM4E (0.43) KDM4ENOS2TLR7HPGDNPC1
SCHEMBL10388599 0.75 KDM4E (0.66) KDM4EALDH1A1HPGDNPC1RAB9A
SCHEMBL10623166 0.74 KDM4E (0.42) KDM4ENOS2TLR7ALDH1A1HPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0714898-B1 PYRAZOLO [1,5-a]PYRIMIDINE DERIVATIVE OTSUKA PHARMA CO LTD (JP) 2001-11-14 EP disclosed
US-5707997-A ANALGESICS OTSUKA PHARMACEUTICAL FACTORY, INC. (JP) 1998-01-13 US disclosed
EP-0714898-A1 PYRAZOLO [1,5-a]PYRIMIDINE DERIVATIVE OTSUKA PHARMACEUTICAL FACTORY, INC. (JP) 1996-06-05 EP disclosed