SCHEMBL8568147

SCHEMBL8568147

CCCCc1cc(Cl)n2nc(C)cc2n1

nearest known ligand 0.41

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
NOS2 P35228 1/20 0.41
TP53 P04637 1/20 0.37
TLR7 Q9NYK1 3/20 0.37
MAOB P27338 1/20 0.35
DPP4 P27487 1/20 0.35
KDM4E B2RXH2 3/20 0.35
ESR1 P03372 1/20 0.34
ESR2 Q92731 1/20 0.34
SMN1; SMN2 Q16637 1/20 0.34
CCNT1 O60563 1/20 0.33
CDK7 P50613 1/20 0.33
CDK9 P50750 1/20 0.33
CCNH P51946 1/20 0.33
NPC1 O15118 1/20 0.33
RAB9A P51151 1/20 0.33
HSD17B10 Q99714 1/20 0.33
USP2 O75604 1/20 0.33
TSHR P16473 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7845874 0.82 KDM4E (0.51) NOS2TP53TLR7MAOBKDM4E
SCHEMBL18780788 0.82 TLR7 (0.42) NOS2TLR7KDM4ESMN1; SMN2NPC1
SCHEMBL18780955 0.77 TLR7 (0.41) NOS2TLR7ESR1ESR2
SCHEMBL7003416 0.76 PDE10A (0.54) NOS2TLR7CCNT1CDK7CDK9
SCHEMBL25465521 0.75 CYP1A2 (0.39) TP53MAOBDPP4KDM4ENPC1
SCHEMBL544920 0.75 RAB9A (0.45) TP53DPP4KDM4ESMN1; SMN2NPC1
SCHEMBL21177636 0.73 KDM4E (0.49) KDM4EESR1ESR2SMN1; SMN2HSD17B10
SCHEMBL1934522 0.73 PDE10A (0.48) TP53MAOBDPP4KDM4ESMN1; SMN2
SCHEMBL545503 0.73 MAOB (0.38) NOS2TP53TLR7MAOBKDM4E
SCHEMBL10626008 0.72 DPP4 (0.42) TP53TLR7MAOBDPP4KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5843951-A Analgesic composition of pyrazolo(1,5-A) pyrimidines OTSUKA PHARMACEUTICAL FACTORY INC. (JP) 1998-12-01 US disclosed
EP-0795555-A1 ANALGESICS OTSUKA PHARMACEUTICAL FACTORY, INC. (JP) 1997-09-17 EP disclosed