SCHEMBL7845940

SCHEMBL7845940

O=c1c2ccc(Br)cc2ccc2cc(Br)ccc12

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ERN1 O75460 1/20 0.50
CYP2A6 P11509 1/20 0.48
HSP90AA1 P07900 1/20 0.46
TLR9 Q9NR96 1/20 0.46
MEN1 O00255 3/20 0.44
KMT2A Q03164 3/20 0.44
MAPT P10636 2/20 0.44
KDM4E B2RXH2 1/20 0.44
ALDH1A1 P00352 1/20 0.44
METAP2 P50579 1/20 0.43
NCEH1 Q6PIU2 2/20 0.42
S100A4 P26447 1/20 0.41
SIRT2 Q8IXJ6 3/20 0.41
SIRT1 Q96EB6 1/20 0.40
BCL2 P10415 1/20 0.39
RXFP1 Q9HBX9 1/20 0.39
CHEK1 O14757 1/20 0.39
AURKA O14965 1/20 0.39
DAPK3 O43293 1/20 0.39
JAK2 O60674 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19871768 0.93 ERN1 (0.46) ERN1CYP2A6HSP90AA1TLR9MEN1
SCHEMBL9068487 0.89 CYP2A6 (0.56) ERN1CYP2A6MEN1KMT2AMAPT
SCHEMBL19862347 0.88 SIRT2 (0.45) ERN1CYP2A6KDM4EALDH1A1NCEH1
SCHEMBL56836 0.84 CYP2A6 (0.57) ERN1CYP2A6MEN1KMT2AMAPT
SCHEMBL16178092 0.82 HSP90AA1 (0.48) ERN1CYP2A6HSP90AA1TLR9MEN1
SCHEMBL12260028 0.81 CYP2A6 (0.55) ERN1CYP2A6MEN1KMT2AMAPT
SCHEMBL646886 0.81 CYP2A6 (0.55) ERN1CYP2A6MEN1KMT2AMAPT
SCHEMBL5342236 0.80 DHODH (0.40) ERN1CYP2A6HSP90AA1TLR9MEN1
SCHEMBL19862341 0.80 TYMS (0.42) ERN1CYP2A6KDM4EALDH1A1SIRT2
SCHEMBL19864880 0.78 HSP90AA1 (0.45) ERN1CYP2A6HSP90AA1TLR9MEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0984963-B1 NOVEL COMPOUNDS ASTRAZENECA AB (SE) 2001-04-11 EP disclosed
US-6162808-A Compounds ASTRAZENECA U.K. LIMITED (GB) 2000-12-19 US disclosed