SCHEMBL9068487

SCHEMBL9068487

O=c1c2ccccc2ccc2cc(Br)ccc12

nearest known ligand 0.64

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP2A6 P11509 2/20 0.56
AKR1B1 P15121 2/20 0.51
MEN1 O00255 1/20 0.49
KMT2A Q03164 1/20 0.49
RXFP1 Q9HBX9 1/20 0.49
MAPK14 Q16539 2/20 0.47
ALDH1A1 P00352 3/20 0.46
HSD17B10 Q99714 2/20 0.46
HIF1A Q16665 1/20 0.46
CYP1B1 Q16678 1/20 0.46
HPRT1 P00492 1/20 0.44
ERN1 O75460 1/20 0.43
TSHR P16473 1/20 0.42
TDP1 Q9NUW8 1/20 0.42
SIRT2 Q8IXJ6 2/20 0.42
PAX8 Q06710 1/20 0.42
MAPT P10636 1/20 0.42
HPGD P15428 1/20 0.42
SIRT1 Q96EB6 1/20 0.41
TDP2 O95551 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9214539 0.90 CYP2A6 (0.52) CYP2A6AKR1B1MEN1KMT2ARXFP1
SCHEMBL7845940 0.89 ERN1 (0.50) CYP2A6MEN1KMT2ARXFP1MAPK14
SCHEMBL19871768 0.88 ERN1 (0.46) CYP2A6AKR1B1MEN1KMT2ARXFP1
SCHEMBL4354069 0.87 CYP2A6 (0.65) CYP2A6MEN1KMT2ARXFP1ALDH1A1
SCHEMBL18646836 0.85 HPRT1 (0.64) CYP2A6MEN1KMT2ARXFP1ALDH1A1
SCHEMBL11179246 0.83 MEN1 (0.49) CYP2A6AKR1B1MEN1KMT2ARXFP1
SCHEMBL9765502 0.80 ALDH1A1 (0.52) CYP2A6AKR1B1MAPK14ALDH1A1HSD17B10
SCHEMBL268735 0.80 ALDH1A1 (0.65) CYP2A6AKR1B1MAPK14ALDH1A1HSD17B10
SCHEMBL30186719 0.80 ALDH1A1 (0.65) CYP2A6AKR1B1MAPK14ALDH1A1HSD17B10
SCHEMBL29391827 0.80 ALDH1A1 (0.65) CYP2A6AKR1B1MAPK14ALDH1A1HSD17B10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 35 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-10693075-B2 Spiro compound and organic electronic device comprising the same SHANGHAI NICHEM FINE CHEMICAL CO., LTD. (CN) 2020-06-23 US disclosed
US-10693075-B2 Spiro compound and organic electronic device comprising the same SHANGHAI NICHEM FINE CHEMICAL CO., LTD. (CN) 2020-06-23 US disclosed
US-10693077-B2 Compound and organic electronic device using the same SHANGHAI NICHEM FINE CHEMICAL CO., LTD. (CN) 2020-06-23 US disclosed
US-10483468-B2 Compound and organic electronic device using the same SHANGHAI NICHEM FINE CHEMICAL CO., LTD. (CN) 2019-11-19 US disclosed
US-10476006-B2 Compound and organic electronic device using the same SHANGHAI NICHEM FINE CHEMICAL CO., LTD. (CN) 2019-11-12 US disclosed
US-10454039-B2 Compound and organic electronic device using the same SHANGHAI NICHEM FINE CHEMICAL CO., LTD. (CN) 2019-10-22 US disclosed
US-10454039-B2 Compound and organic electronic device using the same SHANGHAI NICHEM FINE CHEMICAL CO., LTD. (CN) 2019-10-22 US disclosed
EP-3281936-B1 COMPOUND AND ORGANIC ELECTRONIC DEVICE USING THE SAME SHANGHAI NICHEM FINE CHEMICAL CO LTD (CN) 2019-10-09 EP disclosed
US-10431751-B2 Compound and organic electronic device comprising the same SHANGHAI NICHEM FINE CHEMICAL CO., LTD. (CN) 2019-10-01 US disclosed
US-10424744-B2 Compound and organic electronic device comprising the same SHANGHAI NICHEM FINE CHEMICAL CO., LTD. (CN) 2019-09-24 US disclosed
US-20170279050-A1 COMPOUND AND ORGANIC ELECTRONIC DEVICE USING THE SAME NICHEM FINE TECHNOLOGY CO., LTD. (TW) 2017-09-28 US disclosed
US-20170213971-A1 Novel compound and organic electronic device comprising the same SHANGHAI NICHEM FINE CHEMICAL CO., LTD. (CN) 2017-07-27 US disclosed
US-20170213970-A1 Novel compound and organic electronic device comprising the same SHANGHAI NICHEM FINE CHEMICAL CO., LTD. (CN) 2017-07-27 US disclosed
US-20170213978-A1 COMPOUND AND ORGANIC ELECTRONIC DEVICE USING THE SAME NICHEM FINE TECHNOLOGY CO., LTD. (TW) 2017-07-27 US disclosed
US-5492917-A CARDIOVASCULAR DISORDERS; HYPOTENSIVE, ANTIISCHEMIC,ANTISHOCK, ANTIINFLAMMATORY, ANTIALLERGEN AGENTS MERCK & CO., INC. (US) 1996-02-20 US disclosed
EP-0319073-B1 Cyclo-octane neuroprotective agents MERCK SHARP & DOHME (GB) 1995-08-23 EP disclosed
WO-1995008989-A1 ENDOTHELIN ANTAGONISTS INCORPORATING A CYCLOBUTANE MERCK & CO., INC. (US) 1995-04-06 WO disclosed
EP-0272621-B1 Method for the production of 5H-dibenzo[a,d]cyclohepten-5-ones BASF Aktiengesellschaft (DE) 1991-11-27 EP disclosed
EP-0319073-A2 Cyclo-octane neuroprotective agents MERCK SHARP & DOHME LTD. (GB) 1989-06-07 EP disclosed
EP-0272621-A2 Method for the production of 5H-dibenzo[a,d]cyclohepten-5-ones BASF Aktiengesellschaft (DE) 1988-06-29 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (11 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-10424744-B2 Compound and organic electronic device comprising the same CHRM1, CHRM2, ESR1 CYP2A6 518/4885AKR1B1 1834/4885MEN1 305/4885
US-10693075-B2 Spiro compound and organic electronic device comprising the same ESRRA, REN, ESRRB CYP2A6 632/4885AKR1B1 35/4885MEN1 2448/4885
US-20170213978-A1 COMPOUND AND ORGANIC ELECTRONIC DEVICE USING THE SAME OR51E2, OR10J3, ESR1 CYP2A6 268/4885AKR1B1 2632/4885MEN1 481/4885
US-10693077-B2 Compound and organic electronic device using the same SOD1, SCO2, RCOR3 CYP2A6 1142/4885AKR1B1 496/4885MEN1 2385/4885
US-20170279050-A1 COMPOUND AND ORGANIC ELECTRONIC DEVICE USING THE SAME ESRRA, ESRRB, RCOR3 CYP2A6 902/4885AKR1B1 387/4885MEN1 3217/4885
US-10431751-B2 Compound and organic electronic device comprising the same CHRM1, CHRM2, ESR1 CYP2A6 518/4885AKR1B1 1834/4885MEN1 305/4885
US-10476006-B2 Compound and organic electronic device using the same ESR1, AOC2, PIEZO1 CYP2A6 112/4885AKR1B1 1450/4885MEN1 205/4885
US-20170213970-A1 Novel compound and organic electronic device comprising the same CHRM1, CHRM2, ESR1 CYP2A6 762/4885AKR1B1 1993/4885MEN1 251/4885
US-20170213971-A1 Novel compound and organic electronic device comprising the same CHRM1, CHRM2, ESR1 CYP2A6 762/4885AKR1B1 1993/4885MEN1 251/4885
US-10454039-B2 Compound and organic electronic device using the same ORC3, AOX1, RCOR3 CYP2A6 497/4885AKR1B1 447/4885MEN1 2797/4885
US-10483468-B2 Compound and organic electronic device using the same ORC3, RBX1, CBX3 CYP2A6 1506/4885AKR1B1 920/4885MEN1 1725/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.