SCHEMBL7846356

SCHEMBL7846356

O=C(O)CCCCCOC1CCc2ccccc21

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTR2C P28335 1/20 0.53
SLC6A3 Q01959 1/20 0.53
GPR84 Q9NQS5 2/20 0.45
IDO1 P14902 2/20 0.45
FFAR1 O14842 3/20 0.43
PPARA Q07869 2/20 0.40
MAPT P10636 1/20 0.40
RXFP1 Q9HBX9 1/20 0.40
HDAC3 O15379 1/20 0.40
HDAC4 P56524 1/20 0.40
HDAC1 Q13547 1/20 0.40
HDAC7 Q8WUI4 1/20 0.40
HDAC2 Q92769 1/20 0.40
HDAC10 Q969S8 1/20 0.40
HDAC11 Q96DB2 1/20 0.40
HDAC8 Q9BY41 1/20 0.40
HDAC6 Q9UBN7 1/20 0.40
HDAC9 Q9UKV0 1/20 0.40
HDAC5 Q9UQL6 1/20 0.40
TBXA2R P21731 3/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11025088 0.94 HTR2C (0.49) HTR2CSLC6A3GPR84IDO1FFAR1
SCHEMBL452347 0.80 IDO1 (0.50) GPR84IDO1
SCHEMBL30639030 0.80 IDO1 (0.53) HTR2CSLC6A3GPR84IDO1FFAR1
SCHEMBL2092235 0.80 IDO1 (0.53) HTR2CSLC6A3GPR84IDO1FFAR1
SCHEMBL9626216 0.79 IDO1 (0.51) GPR84IDO1CTSVCTSLCTSS
SCHEMBL448580 0.79 IDO1 (0.51) GPR84IDO1
SCHEMBL449978 0.77 IDO1 (0.53) GPR84IDO1
SCHEMBL19359157 0.76 IDO1 (0.56) GPR84IDO1FFAR1
SCHEMBL7846354 0.76 SLC6A3 (0.46) HTR2CSLC6A3PPARAMAPTRXFP1
SCHEMBL10364010 0.75 ALDH1A1 (0.47) HTR2CSLC6A3GPR84IDO1ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0558677-B1 BIOLOGICALLY ACTIVE AMINES ASTRAZENECA AB (SE) 2001-08-16 EP disclosed
US-5648370-A 7-(2-aminoethyl) benzothiazolones ASTRA PHARMACEUTICALS LIMITED (GB) 1997-07-15 US disclosed
EP-0558677-A1 BIOLOGICALLY ACTIVE AMINES Astra Pharmaceuticals Limited (GB) 1993-09-08 EP disclosed
WO-1992008708-A1 BIOLOGICALLY ACTIVE AMINES FISONS PLC (GB) 1992-05-29 WO disclosed