SCHEMBL7846463

SCHEMBL7846463

Cc1cccc2[nH]c(CCC(=O)Nc3ccc4ccn(CC[C@@H](NC(=O)c5c[nH]cn5)[C@H](C)O)c4c3)nc12

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADA P00813 10/20 0.40
MMP2 P08253 2/20 0.38
MMP9 P14780 2/20 0.38
MMP8 P22894 2/20 0.38
MMP13 P45452 1/20 0.37
TNKS O95271 1/20 0.37
PARP1 P09874 1/20 0.37
TNKS2 Q9H2K2 1/20 0.37
PARP2 Q9UGN5 1/20 0.37
PARP4 Q9UKK3 1/20 0.37
PARP3 Q9Y6F1 1/20 0.37
CYP1A2 P05177 1/20 0.35
CYP3A4 P08684 1/20 0.35
CYP2C19 P33261 1/20 0.35
ALDH1A1 P00352 2/20 0.34
HDAC3 O15379 1/20 0.34
HDAC1 Q13547 1/20 0.34
HDAC6 Q9UBN7 1/20 0.34
USP2 O75604 1/20 0.33
MAPT P10636 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7845268 0.90 ADA (0.41) ADAMMP2MMP9MMP8MMP13
SCHEMBL7845082 0.85 ADA (0.38) ADAMMP2MMP9MMP8MMP13
SCHEMBL7850303 0.77 MMP2 (0.35) ADAMMP2MMP9MMP8MMP13
SCHEMBL7836765 0.77 ADA (0.71) ADA
SCHEMBL7847122 0.75 ADA (0.50) ADAALDH1A1HDAC3HDAC1HDAC6
SCHEMBL7848612 0.73 ADA (0.60) ADAALDH1A1HDAC3HDAC1HDAC6
SCHEMBL7837035 0.72 ADA (0.59) ADAHDAC3HDAC1HDAC6
SCHEMBL7846603 0.68 ADA (0.54) ADAHDAC3HDAC1HDAC6
SCHEMBL7850182 0.67 ADA (0.54) ADA
SCHEMBL7850108 0.65 ADA (0.39) ADAALDH1A1MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1161429-A2 HETEROCYCLIC COMPOUNDS AS ADENOSINE DEAMINASE INHIBITORS FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 2001-12-12 EP disclosed
WO-2000055155-A2 HETEROCYCLIC COMPOUNDS AS ADENOSINE DEAMINASE INHIBITORS FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 2000-09-21 WO disclosed