SCHEMBL7848612

SCHEMBL7848612

Cc1ccc(CCC(=O)Nc2ccc3ccn(CC[C@H](CO)NC(=O)c4c[nH]cn4)c3c2)cc1

nearest known ligand 0.60

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
ADA P00813 12/20 0.60
CNR1 P21554 1/20 0.35
MCHR1 Q99705 1/20 0.34
ALDH1A1 P00352 1/20 0.34
MAPT P10636 1/20 0.34
HDAC3 O15379 1/20 0.34
HDAC1 Q13547 1/20 0.34
HDAC6 Q9UBN7 1/20 0.34
RORC P51449 1/20 0.34
CDK8 P49336 1/20 0.34
ROCK1 Q13464 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7837035 0.87 ADA (0.59) ADAHDAC3HDAC1HDAC6
SCHEMBL7846603 0.84 ADA (0.54) ADAMCHR1HDAC3HDAC1HDAC6
SCHEMBL7850182 0.77 ADA (0.54) ADACNR1MCHR1
SCHEMBL7827408 0.77 CNR1 (0.47) CNR1MAPT
SCHEMBL6936476 0.75 ADA (1.00) ADA
SCHEMBL7836409 0.75 ADA (0.58) ADA
SCHEMBL7847122 0.74 ADA (0.50) ADAMCHR1ALDH1A1MAPTHDAC3
SCHEMBL7850108 0.74 ADA (0.39) ADAALDH1A1MAPT
SCHEMBL7846463 0.73 ADA (0.40) ADAALDH1A1MAPTHDAC3HDAC1
SCHEMBL7845082 0.73 ADA (0.38) ADACNR1ALDH1A1MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1161429-A2 HETEROCYCLIC COMPOUNDS AS ADENOSINE DEAMINASE INHIBITORS FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 2001-12-12 EP disclosed
WO-2000055155-A2 HETEROCYCLIC COMPOUNDS AS ADENOSINE DEAMINASE INHIBITORS FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 2000-09-21 WO disclosed