SCHEMBL7846601

SCHEMBL7846601

COc1ccc(C(=O)C(Br)c2cc(C)cs2)cc1

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.49
CYP1A2 P05177 1/20 0.49
CES2 O00748 1/20 0.41
CES1 P23141 1/20 0.41
NPSR1 Q6W5P4 2/20 0.40
TDP1 Q9NUW8 2/20 0.40
CA2 P00918 5/20 0.40
CA1 P00915 4/20 0.40
RAB9A P51151 3/20 0.40
LMNA P02545 2/20 0.40
GSK3B P49841 1/20 0.40
MEN1 O00255 1/20 0.40
MAPT P10636 1/20 0.40
MAPK1 P28482 1/20 0.40
KMT2A Q03164 1/20 0.40
RXFP1 Q9HBX9 1/20 0.40
PARP1 P09874 1/20 0.39
PARP10 Q53GL7 1/20 0.39
PARP2 Q9UGN5 1/20 0.39
PARP4 Q9UKK3 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7833590 0.87 ALDH1A1 (0.38) ALDH1A1CES2CES1NPSR1TDP1
SCHEMBL7843105 0.84 NPC1 (0.38) CES2CES1TDP1CA2CA1
SCHEMBL7508732 0.83 NPC1 (0.36) ALDH1A1CYP1A2CES2CES1TDP1
SCHEMBL7843947 0.83 CES2 (0.41) ALDH1A1CES2CES1CA2CA1
SCHEMBL7834093 0.77 CES2 (0.41) ALDH1A1CES2CES1TDP1RAB9A
SCHEMBL3105019 0.75 ALDH1A1 (0.55) ALDH1A1CYP1A2CES2CES1NPSR1
SCHEMBL2150940 0.75 ALDH1A1 (0.55) ALDH1A1CYP1A2CES2CES1NPSR1
SCHEMBL11468389 0.74 DAO (0.39) ALDH1A1CYP1A2LMNAMEN1KMT2A
SCHEMBL7847644 0.74 CES2 (0.44) ALDH1A1CYP1A2CES2CES1NPSR1
SCHEMBL3089210 0.74 ALDH1A1 (0.62) ALDH1A1CYP1A2CES2CES1NPSR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1125932-A2 Substituted thiazoles for the treatment of inflammation G.D. SEARLE & CO. (US) 2001-08-22 EP disclosed
US-5668161-A Substituted thiazoles for the treatment of inflammation G.D. SEARLE & CO. (US) 1997-09-16 US disclosed