SCHEMBL7846661

SCHEMBL7846661

COC(=O)c1cccnc1-c1cccc(N(C(=N)NC(=O)OC(C)(C)C)C(=O)OC(C)(C)C)c1

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ATR Q13535 1/20 0.36
ALOX5AP P20292 1/20 0.36
METAP2 P50579 1/20 0.35
PKM P14618 1/20 0.33
L3MBTL1 Q9Y468 1/20 0.33
RORB Q92753 1/20 0.33
TDP1 Q9NUW8 1/20 0.33
BRD4 O60885 1/20 0.32
SLC40A1 Q9NP59 1/20 0.32
F2 P00734 2/20 0.32
F10 P00742 2/20 0.32
PRSS1 P07477 2/20 0.32
PRSS2 P07478 2/20 0.32
PRSS3 P35030 2/20 0.32
FAAH O00519 1/20 0.32
CNR2 P34972 1/20 0.31
TDP2 O95551 1/20 0.31
MAP2K1 Q02750 1/20 0.31
ALOX15 P16050 1/20 0.31
HTT P42858 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7842307 0.87 TRPV1 (0.37) BRD4TDP2
SCHEMBL7847206 0.81 NQO2 (0.34) L3MBTL1BRD4KDM4E
SCHEMBL7847267 0.78 ACACB (0.36) L3MBTL1BRD4HTTALDH1A1
SCHEMBL7846735 0.78 CNR1 (0.40) BRD4
SCHEMBL7232510 0.77 ATR (0.39) ATRALOX5APMETAP2PKML3MBTL1
SCHEMBL7450944 0.75 HPGDS (0.45) KDM4EALDH1A1
SCHEMBL29850324 0.75 NQO2 (0.43) BRD4ALDH1A1
SCHEMBL29597551 0.74 AKT1 (0.39) HTT
SCHEMBL7842830 0.74 CYP17A1 (0.41) ATRALOX5APMETAP2TDP2KDM4E
SCHEMBL7847942 0.73 TDP2 (0.33) TDP2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1157022-A1 PYRIDINE COMPOUNDS AND THEIR PHARMACEUTICAL USE FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 2001-11-28 EP disclosed
WO-2000049015-A1 PYRIDINE COMPOUNDS AND THEIR PHARMACEUTICAL USE FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 2000-08-24 WO disclosed