SCHEMBL7847893

SCHEMBL7847893

CC(C)(C)[Si](C)(C)OC[C@@H](CCc1c[nH]c2ccc(O)cc12)n1cnc(C(N)=O)c1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADA P00813 6/20 0.43
SPR P35270 3/20 0.39
NPSR1 Q6W5P4 4/20 0.39
KDM4E B2RXH2 4/20 0.39
CYP3A4 P08684 3/20 0.39
CYP2D6 P10635 3/20 0.39
ALDH1A1 P00352 3/20 0.39
MAPT P10636 3/20 0.39
CYP1A2 P05177 2/20 0.39
BLM P54132 2/20 0.39
IDO1 P14902 1/20 0.39
HPGD P15428 1/20 0.39
NOTUM Q6P988 1/20 0.39
HTR2C P28335 7/20 0.39
HTR1A P08908 5/20 0.39
HTR2A P28223 5/20 0.39
HTR2B P41595 4/20 0.39
HTR1D P28221 3/20 0.39
TSHR P16473 2/20 0.39
HTR7 P34969 2/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7836809 0.93 ADA (0.43) ADAHTR2CHTR2AHTR2B
SCHEMBL7848925 0.90 ADA (0.44) ADA
SCHEMBL7850190 0.87 ADA (0.43) ADAHPGD
SCHEMBL7846263 0.85 ADA (0.48) ADANPSR1KDM4ECYP3A4CYP2D6
SCHEMBL7848923 0.85 CYP1A2 (0.41) ADASPRNPSR1CYP3A4CYP2D6
SCHEMBL6940660 0.84 ADA (0.58) ADASPR
SCHEMBL7848399 0.83 ADA (0.54) ADAKDM4ECYP3A4CYP2D6MAPT
SCHEMBL7850266 0.83 PTPRA (0.41) ADAMAPTHTR1AHTR1DKMT2A
SCHEMBL7847420 0.83 ADA (0.49) ADAKDM4EALDH1A1MAPTHPGD
SCHEMBL6935332 0.76 ADA (0.57) ADAKDM4EHPGDHTR2AKMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1161429-A2 HETEROCYCLIC COMPOUNDS AS ADENOSINE DEAMINASE INHIBITORS FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 2001-12-12 EP disclosed
WO-2000055155-A2 HETEROCYCLIC COMPOUNDS AS ADENOSINE DEAMINASE INHIBITORS FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 2000-09-21 WO disclosed