SCHEMBL7848403

SCHEMBL7848403

CNS(=O)(=O)c1ccc(C2=C(c3ccccc3)C(=O)C(C)(C)O2)c(Cl)c1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
VCAM1 P19320 1/20 0.39
L3MBTL1 Q9Y468 2/20 0.37
PTGS2 P35354 4/20 0.37
ALDH1A1 P00352 1/20 0.36
MCOLN3 Q8TDD5 1/20 0.36
PTGS1 P23219 2/20 0.35
TNNI3K Q59H18 1/20 0.35
CA12 O43570 1/20 0.35
CA1 P00915 1/20 0.35
CA2 P00918 1/20 0.35
CA3 P07451 1/20 0.35
CA4 P22748 1/20 0.35
CA6 P23280 1/20 0.35
CA5A P35218 1/20 0.35
CA7 P43166 1/20 0.35
CA9 Q16790 1/20 0.35
CA13 Q8N1Q1 1/20 0.35
CA14 Q9ULX7 1/20 0.35
CA5B Q9Y2D0 1/20 0.35
LMNA P02545 2/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6995264 0.87 PTGS2 (0.46) PTGS2ALDH1A1PTGS1
SCHEMBL7843236 0.87 ALDH1A1 (0.38) L3MBTL1PTGS2ALDH1A1MCOLN3PTGS1
SCHEMBL7003146 0.86 PTGS2 (0.42) PTGS2PTGS1CA12CA1CA2
SCHEMBL6998761 0.79 PTGES2 (0.39) PTGS2ALDH1A1PTGS1BRAFPTGES2
SCHEMBL6999198 0.78 PTGS2 (0.32) L3MBTL1PTGS2
SCHEMBL7001429 0.78 PTGS2 (0.48) PTGS2PTGS1
SCHEMBL7001112 0.77 CA1 (0.43) PTGS2PTGS1CA12CA1CA2
SCHEMBL6996726 0.77 PTGS2 (0.43) L3MBTL1PTGS2ALDH1A1PTGS1
SCHEMBL7842902 0.76 MMP1 (0.42) PTGS2PTGS1TNNI3KCA12CA1
SCHEMBL7001462 0.76 PTGS2 (0.49) PTGS2PTGS1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1109799-A1 4,5-DIARYL-3(2H)-FURANONE DERIVATIVES AS CYCLOOXYGENASE-2 INHIBITORS PACIFIC CORPORATION (KR) 2001-06-27 EP disclosed
WO-2000061571-A1 4,5-DIARYL-3(2H)-FURANONE DERIVATIVES AS CYCLOOXYGENASE-2 INHIBITORS PACIFIC CORPORATION (KR) 2000-10-19 WO disclosed