SCHEMBL7848611

SCHEMBL7848611

[CH2]COc1cc(CCCC)nc2ccccc12

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 1/20 0.46
KMT2A Q03164 1/20 0.46
NCF1 P14598 4/20 0.45
KDM4E B2RXH2 1/20 0.45
ABCB11 O95342 1/20 0.44
LMNA P02545 1/20 0.44
CYP1A2 P05177 1/20 0.44
CYP2D6 P10635 1/20 0.44
SCN1A P35498 1/20 0.44
SCN2A Q99250 1/20 0.44
TDP1 Q9NUW8 1/20 0.44
SCN3A Q9NY46 1/20 0.44
PARP1 P09874 1/20 0.42
GABRP O00591 1/20 0.41
GABRD O14764 1/20 0.41
GABRA1 P14867 1/20 0.41
IDO1 P14902 1/20 0.41
GABRB1 P18505 1/20 0.41
GABRG2 P18507 1/20 0.41
GABRB3 P28472 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8673288 0.86 MEN1 (0.48) MEN1KMT2ANCF1KDM4EABCB11
SCHEMBL31587740 0.84 LMNA (0.56) MEN1KMT2AKDM4EABCB11LMNA
SCHEMBL8412379 0.82 AGTR1 (0.48) MEN1KMT2ANCF1KDM4EABCB11
SCHEMBL21166292 0.80 AGTR1 (0.47) MEN1KMT2ANCF1KDM4ELMNA
SCHEMBL19732877 0.80 AGTR1 (0.47) MEN1KMT2ANCF1KDM4ELMNA
SCHEMBL951984 0.80 LMNA (0.55) MEN1KMT2AKDM4ELMNA
SCHEMBL8410524 0.79 MEN1 (0.43) MEN1KMT2AKDM4EABCB11LMNA
SCHEMBL8671748 0.78 MEN1 (0.51) MEN1KMT2AKDM4EABCB11LMNA
SCHEMBL9179529 0.77 MEN1 (0.53) MEN1KMT2AKDM4EABCB11LMNA
SCHEMBL7838473 0.77 NR1H4 (0.49) KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0498723-B1 Nitrogen containing bicycle compounds, method for their preparation, their use as pharmaceutical and compositions containing them AVENTIS PHARMA SA (FR) 2001-09-19 EP disclosed
EP-0498723-A1 Nitrogen containing bicycle compounds, method for their preparation, their use as pharmaceutical and compositions containing them ROUSSEL UCLAF (FR) 1992-08-12 EP disclosed