SCHEMBL7848819

SCHEMBL7848819

CC(Cc1c[nH]c2ccccc12)C(=O)NC1CCc2ccccc21

nearest known ligand 0.68

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
MMP2 P08253 2/20 0.68
MMP3 P08254 2/20 0.68
MMP9 P14780 2/20 0.68
MMP8 P22894 2/20 0.68
TAOK1 Q7L7X3 3/20 0.56
TAOK3 Q9H2K8 2/20 0.55
POLB P06746 2/20 0.54
KDM4E B2RXH2 1/20 0.54
APAF1 O14727 1/20 0.54
MAPT P10636 1/20 0.54
RECQL P46063 1/20 0.54
L3MBTL1 Q9Y468 1/20 0.54
ECE1 P42892 9/20 0.54
NMBR P28336 2/20 0.52
CTDSP1 Q9GZU7 1/20 0.51

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14261304 0.82 MMP2 (0.57) MMP2MMP3MMP9MMP8MAPT
SCHEMBL5652426 0.82 TAOK1 (0.60) MMP2MMP3MMP9MMP8TAOK1
SCHEMBL31730289 0.82 TAOK1 (0.60) MMP2MMP3MMP9MMP8TAOK1
SCHEMBL5653439 0.82 TAOK1 (0.60) MMP2MMP3MMP9MMP8TAOK1
SCHEMBL7854930 0.81 POLB (0.60) MMP2MMP3MMP9MMP8POLB
SCHEMBL7846847 0.80 HPGD (0.67) MMP2MMP3MMP9MMP8MAPT
SCHEMBL7675962 0.79 MMP2 (0.63) MMP2MMP9MMP8POLBKDM4E
SCHEMBL14261305 0.78 HPGD (0.58) MMP2MMP3MMP9MMP8KDM4E
SCHEMBL24105928 0.78 MMP2 (0.48) MMP2MMP3MMP9MMP8TAOK1
SCHEMBL9268039 0.77 NMBR (0.65) NMBR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1140914-A1 NON-PEPTIDE NK1 RECEPTORS ANTAGONISTS WARNER-LAMBERT COMPANY (US) 2001-10-10 EP disclosed
WO-2000037462-A1 NON-PEPTIDE NK1 RECEPTORS ANTAGONISTS WARNER-LAMBERT COMPANY (US) 2000-06-29 WO disclosed