SCHEMBL7848965

SCHEMBL7848965

COc1ccc(C(N)=O)cc1N1CCN2CCC1C2

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPK1 P28482 1/20 0.41
PDE4D Q08499 2/20 0.41
PDE4A P27815 1/20 0.41
PDE4B Q07343 1/20 0.41
PDE4C Q08493 1/20 0.41
ALDH1A1 P00352 4/20 0.40
PKM P14618 2/20 0.40
HPGD P15428 1/20 0.40
HSD17B10 Q99714 1/20 0.40
MKNK1 Q9BUB5 1/20 0.39
MKNK2 Q9HBH9 1/20 0.39
KDM4E B2RXH2 2/20 0.39
LMNA P02545 1/20 0.39
GAA P10253 1/20 0.38
SLC2A1 P11166 1/20 0.38
SLC2A2 P11168 1/20 0.38
SLC2A3 P11169 1/20 0.38
CYP2D6 P10635 1/20 0.38
MAPT P10636 1/20 0.38
HTR1D P28221 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7848968 0.81 MAPT (0.47) MAPK1ALDH1A1KDM4ELMNAGAA
SCHEMBL6355486 0.74 CTPS1 (0.58) MAPK1PDE4DPDE4APDE4BPDE4C
Hydrochloric Acid SCHEMBL6353867 0.73 CTPS1 (0.57) MAPK1PDE4DPDE4APDE4BPDE4C
SCHEMBL1397384 0.70 KDM4E (0.63) ALDH1A1HSD17B10KDM4ESLC2A1SLC2A2
SCHEMBL7845695 0.70 MAPK1 (0.48) MAPK1PDE4DPDE4APDE4BPDE4C
SCHEMBL2779632 0.69 HTR3A (0.59) MAPK1LMNASLC2A1SLC2A2SLC2A3
Hydrochloric Acid SCHEMBL6343776 0.69 KDM4E (0.62) ALDH1A1HSD17B10KDM4ESLC2A1SLC2A2
Hydrochloric Acid SCHEMBL3072094 0.69 KDM4E (0.62) ALDH1A1HSD17B10KDM4ESLC2A1SLC2A2
SCHEMBL7835719 0.69 CHRNA4 (0.47) MAPK1PDE4DPDE4APDE4BPDE4C
SCHEMBL7035600 0.69 OPRK1 (0.49) MAPK1SLC2A1SLC2A2SLC2A3HTR1D

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1066288-A2 NOVEL COMPOUNDS SMITHKLINE BEECHAM PLC (GB) 2001-01-10 EP disclosed
WO-1999042465-A2 SULPHONAMIDE DERIVATIVES BEING 5-HT6 RECEPTOR ANTAGONISTS AND PROCESS FOR THEIR PREPARATION SMITHKLINE BEECHAM PLC (GB) 1999-08-26 WO disclosed