SCHEMBL7849294

SCHEMBL7849294

COC(=O)C=CCC(CCC#N)(c1ccccc1)c1ccccc1

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
POLB P06746 1/20 0.36
RAB9A P51151 1/20 0.36
KCNN4 O15554 1/20 0.36
ALDH1A1 P00352 5/20 0.35
MAPT P10636 5/20 0.35
KDM4E B2RXH2 2/20 0.34
KMT2A Q03164 1/20 0.34
SMN1; SMN2 Q16637 1/20 0.34
TTR P02766 1/20 0.34
APP P05067 1/20 0.34
LMNA P02545 3/20 0.34
GAA P10253 1/20 0.34
CA12 O43570 1/20 0.33
CA1 P00915 1/20 0.33
CA2 P00918 1/20 0.33
TYR P14679 1/20 0.33
CA7 P43166 1/20 0.33
CA9 Q16790 1/20 0.33
CA14 Q9ULX7 1/20 0.33
TP53 P04637 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7849292 1.00 POLB (0.36) POLBRAB9AKCNN4ALDH1A1MAPT
SCHEMBL7848935 0.74 ALDH1A1 (0.34) ALDH1A1MAPTGAAKCNA3HTT
SCHEMBL7847690 0.74 LMNA (0.40) POLBKCNN4ALDH1A1MAPTKDM4E
SCHEMBL7465712 0.70 ALDH1A1 (0.39) POLBALDH1A1MAPTKDM4EKMT2A
SCHEMBL7706699 0.69 KIF11 (0.50) RAB9AALDH1A1MAPTKDM4EKMT2A
SCHEMBL7706702 0.69 KIF11 (0.50) RAB9AALDH1A1MAPTKDM4EKMT2A
SCHEMBL7816354 0.68 SMN1; SMN2 (0.47) POLBALDH1A1MAPTKMT2ASMN1; SMN2
SCHEMBL4799716 0.67 HCAR2 (0.46) POLBRAB9AALDH1A1MAPTKMT2A
SCHEMBL4799720 0.67 HCAR2 (0.46) POLBRAB9AALDH1A1MAPTKMT2A
SCHEMBL7824378 0.67 MEN1 (0.42) POLBRAB9AALDH1A1MAPTKMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1129076-A1 TETRAHYDROISOQUINOLINE DERIVATIVES AS LHRH ANTAGONISTS ABBOTT LABORATORIES (US) 2001-09-05 EP disclosed
WO-2000029380-A1 TETRAHYDROISOQUINOLINE DERIVATIVES AS LHRH ANTAGONISTS ABBOTT LABORATORIES (US) 2000-05-25 WO disclosed
US-5981521-A USEFUL FOR TREATING VARIOUS HORMONE DEPENDENT DISEASES, INCLUDING PROSTATE CANCER, ENDOMETRIOSIS, UTERINE FIBROIDS, PRECOCIOUS PUBERTY, BENIGN PROSTATE HYPERTROPY AND IN VITRO FERTILIZATION ABBOTT LABORATORIES (US) 1999-11-09 US disclosed