SCHEMBL7849465

SCHEMBL7849465

Cn1c(C(=O)O)c(-c2ccc(F)cc2)c2cccnc2c1=O

nearest known ligand 0.63

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
TACR1 P25103 14/20 0.63
MAPK14 Q16539 4/20 0.44
GRIA2 P42262 1/20 0.42
GRIA4 P48058 1/20 0.42
AHR P35869 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7841672 0.90 TACR1 (0.52) TACR1MAPK14GRIA2GRIA4
SCHEMBL7850487 0.90 TACR1 (0.59) TACR1GRIA2GRIA4
SCHEMBL7851995 0.89 TACR1 (0.62) TACR1MAPK14AHR
SCHEMBL7852137 0.89 TACR1 (0.56) TACR1
Hydrochloric Acid SCHEMBL7852820 0.88 TACR1 (0.66) TACR1GRIA2GRIA4
SCHEMBL7850928 0.86 TACR1 (0.47) TACR1MAPK14GRIA2GRIA4
SCHEMBL7849658 0.86 TACR1 (0.54) TACR1GRIA2GRIA4
SCHEMBL7849923 0.83 TACR1 (0.59) TACR1
SCHEMBL7851972 0.82 TACR1 (0.81) TACR1
SCHEMBL8948131 0.82 TACR1 (0.55) TACR1MAPK14GRIA2GRIA4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0652218-B1 Heterocyclic compounds, their production and use TAKEDA CHEMICAL INDUSTRIES LTD (JP) 2001-07-11 EP disclosed
US-5585385-A USEFUL IN TREATING DISORDERS OF MICTURITION; ADMINISTERING TO INHIBIT PLASMA EXTRAVASATION TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1996-12-17 US disclosed
EP-0652218-A1 Heterocyclic compounds, their production and use Takeda Chemical Industries, Ltd. (JP) 1995-05-10 EP disclosed