SCHEMBL7849658

SCHEMBL7849658

COc1ccc(-c2c(C(=O)O)n(C)c(=O)c3ncccc23)cc1

nearest known ligand 0.54

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
TACR1 P25103 13/20 0.54
GRIA2 P42262 1/20 0.45
GRIA4 P48058 1/20 0.45
KMT2A Q03164 2/20 0.42
MEN1 O00255 1/20 0.42
KAT2B Q92831 1/20 0.42
KDM4E B2RXH2 1/20 0.42
USP2 O75604 1/20 0.42
ALDH1A1 P00352 1/20 0.42
HPGD P15428 1/20 0.42
HSD17B10 Q99714 1/20 0.42
SLC11A2 P49281 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7852343 0.90 TACR1 (0.53) TACR1KMT2AKAT2BKDM4EUSP2
SCHEMBL7850487 0.88 TACR1 (0.59) TACR1GRIA2GRIA4KMT2AKDM4E
SCHEMBL7852137 0.87 TACR1 (0.56) TACR1KAT2BKDM4EHPGD
Hydrochloric Acid SCHEMBL7852820 0.86 TACR1 (0.66) TACR1GRIA2GRIA4
SCHEMBL7849465 0.86 TACR1 (0.63) TACR1GRIA2GRIA4
SCHEMBL7855252 0.79 TACR1 (0.43) TACR1KMT2AMEN1KAT2BKDM4E
Hydrochloric Acid SCHEMBL7852917 0.78 TACR1 (0.52) TACR1GRIA2GRIA4KMT2A
SCHEMBL7854807 0.78 TACR1 (0.48) TACR1GRIA2GRIA4KMT2AKDM4E
SCHEMBL6636299 0.77 PADI4 (0.47) KMT2AKAT2BKDM4EUSP2ALDH1A1
SCHEMBL7850548 0.76 TACR1 (0.63) TACR1KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0652218-B1 Heterocyclic compounds, their production and use TAKEDA CHEMICAL INDUSTRIES LTD (JP) 2001-07-11 EP disclosed
US-5585385-A USEFUL IN TREATING DISORDERS OF MICTURITION; ADMINISTERING TO INHIBIT PLASMA EXTRAVASATION TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1996-12-17 US disclosed
EP-0652218-A1 Heterocyclic compounds, their production and use Takeda Chemical Industries, Ltd. (JP) 1995-05-10 EP disclosed