SCHEMBL7849572

SCHEMBL7849572

COc1ccc2c(c1OC)NC(=O)C(N)C2

nearest known ligand 0.46

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
ACHE P22303 2/20 0.46
AADAT Q8N5Z0 4/20 0.44
ADRA1A P35348 2/20 0.41
KYAT3 Q6YP21 2/20 0.41
KYAT1 Q16773 1/20 0.41
KDM4E B2RXH2 1/20 0.40
LMNA P02545 1/20 0.40
PARP1 P09874 1/20 0.38
NPC1 O15118 4/20 0.37
RAB9A P51151 4/20 0.37
POLB P06746 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7835962 0.72 GAA (0.43) ACHEKDM4EPOLB
SCHEMBL4070986 0.71 SRC (0.42) ACHEAADATKYAT3
Hydrochloric Acid SCHEMBL7420949 0.70 SRC (0.41) ACHEAADATKYAT3
SCHEMBL8542873 0.68 ADRA1A (0.63) ACHEADRA1ALMNAPOLB
Hydrochloric Acid SCHEMBL9432424 0.68 AADAT (0.47) AADATKYAT3KYAT1
SCHEMBL13007381 0.67 ANPEP (0.40) AADATKYAT3KYAT1
Hydrochloric Acid SCHEMBL9696131 0.67 ADRA1A (0.61) ACHEADRA1ALMNAPOLB
Hydrochloric Acid SCHEMBL2841681 0.66 ANPEP (0.42) AADATKYAT3KYAT1
SCHEMBL12569201 0.66 AADAT (0.39) ACHEAADATPOLB
SCHEMBL4795933 0.66 AADAT (0.52) ACHEAADATADRA1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0802922-B1 NOVEL AMINO ACID DERIVATIVES, METHOD OF PRODUCING THEM AND PHARMACEUTICAL COMPOSITIONS CONTAINING THESE COMPOUNDS BOEHRINGER INGELHEIM PHARMA (DE) 2001-09-26 EP disclosed
EP-0802922-A1 NOVEL AMINO ACID DERIVATIVES, METHOD OF PRODUCING THEM AND PHARMACEUTICAL COMPOSITIONS CONTAINING THESE COMPOUNDS BOEHRINGER INGELHEIM KG (DE) 1997-10-29 EP disclosed
WO-1995023810-A1 NOVEL AMINO ACID DERIVATIVES, METHOD OF PRODUCING THEM AND PHARMACEUTICAL COMPOSITIONS CONTAINING THESE COMPOUNDS BOEHRINGER INGELHEIM KG (DE) 1995-09-08 WO disclosed