SCHEMBL7835962

SCHEMBL7835962

COc1ccc2c(c1OC)NC(=O)C(NC(=O)OC(C)(C)C)C2

nearest known ligand 0.43

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
GAA P10253 2/20 0.43
KDM4E B2RXH2 2/20 0.40
ALDH1A1 P00352 2/20 0.40
POLB P06746 1/20 0.40
HSD17B10 Q99714 1/20 0.40
EPHX2 P34913 1/20 0.40
ACHE P22303 2/20 0.37
NFKB1 P19838 1/20 0.37
NFKB2 Q00653 1/20 0.37
RELA Q04206 1/20 0.37
PLG P00747 1/20 0.36
PDE4B Q07343 2/20 0.36
KDM4D Q6B0I6 1/20 0.36
DDB1 Q16531 1/20 0.34
CRBN Q96SW2 1/20 0.34
CFTR P13569 1/20 0.34
DRD2 P14416 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7835958 0.78 GAA (0.46) GAAKDM4EALDH1A1EPHX2NFKB1
SCHEMBL2842186 0.77 EPHX2 (0.46) GAAEPHX2NFKB1NFKB2RELA
SCHEMBL26518869 0.76 GAA (0.40) GAAKDM4EALDH1A1EPHX2NFKB1
SCHEMBL4806148 0.73 EPHX2 (0.63) GAAEPHX2NFKB1NFKB2RELA
SCHEMBL651277 0.73 EPHX2 (0.63) GAAEPHX2NFKB1NFKB2RELA
SCHEMBL651278 0.73 EPHX2 (0.63) GAAEPHX2NFKB1NFKB2RELA
SCHEMBL29900496 0.73 EPHX2 (0.63) GAAEPHX2NFKB1NFKB2RELA
SCHEMBL2840913 0.72 GAA (0.41) GAAALDH1A1HSD17B10EPHX2PLG
SCHEMBL7849572 0.72 ACHE (0.46) KDM4EPOLBACHE
SCHEMBL7420752 0.72 PYGL (0.47) GAAEPHX2NFKB1NFKB2RELA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0802922-B1 NOVEL AMINO ACID DERIVATIVES, METHOD OF PRODUCING THEM AND PHARMACEUTICAL COMPOSITIONS CONTAINING THESE COMPOUNDS BOEHRINGER INGELHEIM PHARMA (DE) 2001-09-26 EP disclosed
EP-0802922-A1 NOVEL AMINO ACID DERIVATIVES, METHOD OF PRODUCING THEM AND PHARMACEUTICAL COMPOSITIONS CONTAINING THESE COMPOUNDS BOEHRINGER INGELHEIM KG (DE) 1997-10-29 EP disclosed
WO-1995023810-A1 NOVEL AMINO ACID DERIVATIVES, METHOD OF PRODUCING THEM AND PHARMACEUTICAL COMPOSITIONS CONTAINING THESE COMPOUNDS BOEHRINGER INGELHEIM KG (DE) 1995-09-08 WO disclosed