SCHEMBL7853010

SCHEMBL7853010

COc1cccc(B2OB(c3cccc(OC)c3)OB(c3cccc(OC)c3)O2)c1

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ACHE P22303 1/20 0.48
CA1 P00915 1/20 0.47
CA2 P00918 1/20 0.47
CA7 P43166 1/20 0.47
CA9 Q16790 1/20 0.47
ALDH1A1 P00352 1/20 0.47
CYP3A4 P08684 1/20 0.47
CES2 O00748 1/20 0.42
CES1 P23141 1/20 0.42
ENPP2 Q13822 1/20 0.42
CHRM5 P08912 1/20 0.41
CA4 P22748 1/20 0.41
IDO1 P14902 2/20 0.40
AGXT P21549 2/20 0.40
NPC1 O15118 1/20 0.40
RAB9A P51151 1/20 0.40
PARP1 P09874 1/20 0.40
RELA Q04206 1/20 0.40
SMN1; SMN2 Q16637 1/20 0.40
DYRK1A Q13627 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14985998 0.85 NPC1 (0.47) ALDH1A1CHRM5NPC1RAB9ARELA
SCHEMBL14985997 0.82 ACHE (0.44) ACHECA1CA2CA7CA9
SCHEMBL422395 0.81 LPL (0.49) ACHECA1CA2CA7CA9
SCHEMBL6826334 0.80 ACHE (0.41) ACHECA1CA2CA7CA9
SCHEMBL17421920 0.80 ACHE (0.41) ACHECA1CA2CA7CA9
SCHEMBL19417354 0.77 SNCA (0.49) ACHECA1CA2CA7CA9
SCHEMBL14985985 0.75 KCNH2 (0.40) ALDH1A1GAA
1,3-Dimethoxybenzene SCHEMBL9350 0.74 ACHE (0.70) ACHECA1CA2CA7CA9
1,3-Dimethoxybenzene SCHEMBL901285 0.74 ACHE (0.70) ACHECA1CA2CA7CA9
SCHEMBL7858694 0.73 CA1 (0.55) ACHECA1CA2CA7CA9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 9 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9556108-B2 Process for preparing substituted phenylalkanes MALLINCKRODT LLC (US) 2017-01-31 US disclosed
US-9556108-B2 Process for preparing substituted phenylalkanes MALLINCKRODT LLC (US) 2017-01-31 US disclosed
US-20160009635-A1 PROCESS FOR PREPARING SUBSTITUTED PHENYLALKANES MALLINCKRODT PHARMA IP TRADING UNLIMITED COMPANY 2016-01-14 US disclosed
WO-2016007823-A1 PROCESS FOR PREPARING SUBSTITUTED PHENYLALKANES MALLINCKRODT LLC (US) 2016-01-14 WO disclosed
US-20160009635-A1 PROCESS FOR PREPARING SUBSTITUTED PHENYLALKANES MALLINCKRODT PHARMA IP TRADING UNLIMITED COMPANY 2016-01-14 US disclosed
EP-0736509-B1 Processes for preparing optically active alcohols and optically active amines SUMITOMO CHEMICAL CO (JP) 2001-11-14 EP disclosed
US-6025531-A REACTING A PROCHIRAL KETONE WITH A MIXTURE BORON-CONTAINING COMPOUNDS HAVING A BORANE REACTION PRODUCT FROM OPTICALLY ACTIVE BETA-AMINOALCOHOL AND A BORON HYDRIDE OR A METAL BOROHYDRIDE, AND AN OPTICALLY ACTIVE OXAZABOROLIDINE SUMITOMO CHEMICAL COMPANY, LIMITED (JP) 2000-02-15 US disclosed
US-5801280-A Processes for preparing optically active alcohols and optically active amines SUMITOMO CHEMICAL COMPANY, LIMITED (JP) 1998-09-01 US disclosed
EP-0736509-A2 Processes for preparing optically active alcohols and optically active amines SUMITOMO CHEMICAL COMPANY, LIMITED (JP) 1996-10-09 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20160009635-A1 PROCESS FOR PREPARING SUBSTITUTED PHENYLALKANES CYP2E1, CYP1B1, CYP4B1 ACHE 219/4885CA1 3774/4885CA2 2374/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.