SCHEMBL7854059

SCHEMBL7854059

O=C(NC1CCCCC1)C(=O)C1CCCN1C(=O)[C@H](Cc1ccccc1)NC(=O)c1ccc(CN2CCOCC2)cc1

nearest known ligand 0.57

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 1/20 0.57
RAB9A P51151 1/20 0.57
KMT2A Q03164 1/20 0.57
SMN1; SMN2 Q16637 1/20 0.57
KDM4E B2RXH2 1/20 0.55
ACE P12821 13/20 0.49
ACE2 Q9BYF1 6/20 0.49
TSHR P16473 1/20 0.49
ALDH1A1 P00352 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL7856176 0.99 NPC1 (0.56) NPC1RAB9AKMT2ASMN1; SMN2KDM4E
SCHEMBL7845289 0.88 ACE (0.59) ACEACE2TSHR
SCHEMBL7845317 0.86 KMT2A (0.57) NPC1RAB9AKMT2ASMN1; SMN2KDM4E
SCHEMBL7844672 0.83 HTRA1 (0.52) ACEACE2TSHR
SCHEMBL7844467 0.82 NPC1 (0.65) NPC1RAB9AKMT2ASMN1; SMN2KDM4E
SCHEMBL7855038 0.81 KDM4E (0.58) RAB9AKDM4EACEACE2ALDH1A1
SCHEMBL7856866 0.80 ACE (0.55) ACEACE2TSHR
SCHEMBL7852243 0.80 FAP (0.49) ACEACE2ALDH1A1
SCHEMBL7844481 0.80 PKM (0.53) NPC1ACEACE2TSHR
SCHEMBL7845347 0.80 PKM (0.53) NPC1ACEACE2TSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0709373-B1 PYRROLIDINE DERIVATIVE ZAIDAN HOJIN BISEIBUTSU (JP) 2001-10-17 EP disclosed
US-5965556-A KETO-ACID AMIDE DERIVATIVES, PHARMACEUTICAL COMPOSITIONS CONTAINING THEM AND METHODS FOR INHIBITING THE ACTIVITY OF SERINE PROTEASE OR THIOL PROTEASE BY ADMINISTERING THE DERIVATIVE TO A MAMMAL; ALZHEIMER'S DISEASE ZAIDAN HOJIN BISEIBUTSU KAGAKU KENKYUKAI (JP) 1999-10-12 US disclosed
US-5756763-A ENZYME INHIBITOR ZAIDAN HOJIN BISEIBUTSU KAGAKU KENKYUKAI (JP) 1998-05-26 US disclosed
EP-0709373-A1 NOVEL PYRROLIDINE DERIVATIVE ZAIDAN HOJIN BISEIBUTSU KAGAKU KENKYU KAI (JP) 1996-05-01 EP disclosed