SCHEMBL7854615

SCHEMBL7854615

O=C(c1ccc(Cl)cc1)N1CCc2c([nH]c3ccc(Cl)cc23)C1C1(C(=O)O)CCC1

nearest known ligand 0.52

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
KIF11 P52732 3/20 0.52
ALDH1A1 P00352 1/20 0.52
ABCG2 Q9UNQ0 7/20 0.51
SIRT1 Q96EB6 7/20 0.50
ABCB1 P08183 3/20 0.49
MAPKAPK2 P49137 1/20 0.45
SIRT2 Q8IXJ6 3/20 0.44
SIRT3 Q9NTG7 2/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7843919 0.95 ABCG2 (0.55) KIF11ALDH1A1ABCG2SIRT1ABCB1
SCHEMBL7855327 0.93 KIF11 (0.47) KIF11ALDH1A1ABCG2SIRT1ABCB1
SCHEMBL7852589 0.92 ABCG2 (0.55) KIF11ALDH1A1ABCG2SIRT1ABCB1
SCHEMBL7853658 0.89 SIRT1 (0.46) KIF11ALDH1A1ABCG2SIRT1ABCB1
SCHEMBL7680030 0.88 SIRT1 (0.62) KIF11SIRT1MAPKAPK2SIRT2SIRT3
SCHEMBL7855042 0.88 ABCG2 (0.45) KIF11ALDH1A1ABCG2SIRT1ABCB1
SCHEMBL7847564 0.87 SIRT1 (0.47) KIF11ABCG2SIRT1ABCB1MAPKAPK2
SCHEMBL7680379 0.87 MAPT (0.51) KIF11ALDH1A1ABCG2SIRT1ABCB1
SCHEMBL7853788 0.86 SIRT1 (0.46) KIF11ABCG2SIRT1ABCB1MAPKAPK2
SCHEMBL7852116 0.86 NPSR1 (0.56) KIF11ABCG2SIRT1ABCB1MAPKAPK2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1070716-A1 Beta-carboline derivatives, process for their preparation and pharmaceutical compositions containing them ADIR ET COMPAGNIE (FR) 2001-01-24 EP disclosed