Benzamide

Benzamide

SCHEMBL7855950

NC(=O)c1ccc(-c2ccnc(NCC(c3ccccc3)c3ccccc3)n2)cc1.NC(=O)c1ccc(-c2ccnc(NCc3cccc(C(F)(F)F)c3)n2)cc1.NC(=O)c1ccccc1

nearest known ligand 0.49

Full drug profile on Sugi Atlas →

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
VNN1 O95497 2/20 0.49
CAMKK2 Q96RR4 5/20 0.48
MAPK8 P45983 3/20 0.48
GSK3B P49841 2/20 0.48
PIK3CG P48736 2/20 0.48
AURKA O14965 3/20 0.46
RPS6KB1 P23443 1/20 0.46
AURKB Q96GD4 1/20 0.46
MAPK10 P53779 1/20 0.46
HDAC1 Q13547 2/20 0.43
HDAC3 O15379 1/20 0.43
HDAC2 Q92769 1/20 0.43
HDAC6 Q9UBN7 1/20 0.43
MAOB P27338 1/20 0.43
GPR52 Q9Y2T5 1/20 0.43
MAPK14 Q16539 2/20 0.42
EPHX1 P07099 1/20 0.42
BCHE P06276 1/20 0.42
TRPM8 Q7Z2W7 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5093362 0.90 VNN1 (0.55) VNN1CAMKK2MAPK8GSK3BPIK3CG
SCHEMBL5094134 0.86 CAMKK2 (0.54) VNN1CAMKK2MAPK8GSK3BPIK3CG
SCHEMBL5092162 0.84 MAPK8 (0.61) CAMKK2MAPK8GSK3BPIK3CGMAPK10
SCHEMBL5100707 0.81 CAMKK2 (0.49) VNN1CAMKK2MAPK8GSK3BPIK3CG
SCHEMBL5100280 0.79 HDAC1 (0.53) VNN1CAMKK2MAPK8GSK3BPIK3CG
SCHEMBL27576350 0.77 CAMKK2 (0.55) CAMKK2MAPK8GSK3BPIK3CGMAPK10
SCHEMBL5094793 0.76 MAPK8 (0.58) CAMKK2MAPK8GSK3BPIK3CGMAPK10
SCHEMBL5094438 0.76 CAMKK2 (0.54) VNN1CAMKK2MAPK8GSK3BPIK3CG
SCHEMBL5100273 0.76 CAMK2D (0.55) VNN1CAMKK2MAPK8GSK3BPIK3CG
SCHEMBL5091408 0.76 CAMKK2 (0.54) CAMKK2MAPK8GSK3BPIK3CGAURKA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1087963-A1 INHIBITORS OF GLYCOGEN SYNTHASE KINASE 3 Chiron Corporation (US) 2001-04-04 EP disclosed
WO-1999065897-A1 INHIBITORS OF GLYCOGEN SYNTHASE KINASE 3 CHIRON CORPORATION (US) 1999-12-23 WO disclosed