SCHEMBL7859537

SCHEMBL7859537

CS(=O)(=O)Nc1cc2occ(NC=O)c(=O)c2cc1Nc1ccc(F)cc1F

nearest known ligand 0.56

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
PTGS1 P23219 3/20 0.56
ADORA3 P0DMS8 1/20 0.56
MIF P14174 1/20 0.56
PDE4A P27815 1/20 0.56
PDE4D Q08499 1/20 0.56
PTGS2 P35354 4/20 0.48
PLA2G7 Q13093 4/20 0.38
PTPN1 P18031 1/20 0.36
KMT2A Q03164 1/20 0.33
SOS1 Q07889 1/20 0.33
MAPK14 Q16539 1/20 0.32
BRD4 O60885 1/20 0.32
KIT P10721 1/20 0.32
TSHR P16473 1/20 0.31
HSD17B10 Q99714 1/20 0.31
ALDH1A1 P00352 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7859528 0.89 ADORA3 (0.63) PTGS1ADORA3MIFPDE4APDE4D
SCHEMBL7859555 0.81 PTGS2 (0.48) PTGS1ADORA3MIFPDE4APDE4D
SCHEMBL10334608 0.78 PTGS1 (0.76) PTGS1ADORA3MIFPDE4APDE4D
SCHEMBL30842776 0.74 PTGS1 (0.70) PTGS1ADORA3MIFPDE4APDE4D
SCHEMBL29377983 0.73 ADORA3 (0.69) PTGS1ADORA3MIFPDE4APDE4D
SCHEMBL29377471 0.73 ADORA3 (0.69) PTGS1ADORA3MIFPDE4APDE4D
SCHEMBL10415468 0.73 ADORA3 (0.78) PTGS1ADORA3MIFPDE4APDE4D
Iguratimod SCHEMBL26326 0.72 PTGS1 (1.00) PTGS1ADORA3MIFPDE4APDE4D
Iguratimod SCHEMBL29366981 0.72 PTGS1 (1.00) PTGS1ADORA3MIFPDE4APDE4D
Potassium SCHEMBL29375000 0.72 ADORA3 (0.68) PTGS1ADORA3MIFPDE4APDE4D

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 8 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0695547-B1 IMMUNOMODULATOR, CELL ADHESION INHIBITOR, AND AGENT FOR TREATING AND PREVENTING AUTOIMMUNE DISEASES TOYAMA CHEMICAL CO LTD (JP) 2001-08-08 EP claimed
US-6166068-A Immunomodulator, cell adhesion inhibitor, and agent for treating, and preventing autoimmune diseases TOYAMA CHEMICAL CO., LTD. (JP) 2000-12-26 US claimed
US-5922755-A ADMINSTERING 4H-1-BENZOPYRAN-4-ONE DERIVATIVE TOYAMA CHEMICAL CO., LTD. (JP) 1999-07-13 US claimed
EP-0695547-A1 IMMUNOMODULATOR, CELL ADHESION INHIBITOR, AND AGENT FOR TREATING AND PREVENTING AUTOIMMUNE DISEASES TOYAMA CHEMICAL CO., LTD. (JP) 1996-02-07 EP claimed
EP-0695547-B1 IMMUNOMODULATOR, CELL ADHESION INHIBITOR, AND AGENT FOR TREATING AND PREVENTING AUTOIMMUNE DISEASES TOYAMA CHEMICAL CO LTD (JP) 2001-08-08 EP disclosed
US-6166068-A Immunomodulator, cell adhesion inhibitor, and agent for treating, and preventing autoimmune diseases TOYAMA CHEMICAL CO., LTD. (JP) 2000-12-26 US disclosed
US-5922755-A ADMINSTERING 4H-1-BENZOPYRAN-4-ONE DERIVATIVE TOYAMA CHEMICAL CO., LTD. (JP) 1999-07-13 US disclosed
EP-0695547-A1 IMMUNOMODULATOR, CELL ADHESION INHIBITOR, AND AGENT FOR TREATING AND PREVENTING AUTOIMMUNE DISEASES TOYAMA CHEMICAL CO., LTD. (JP) 1996-02-07 EP disclosed