SCHEMBL7860146

SCHEMBL7860146

CCCNCCC.O=S(=O)(Cc1ccc2c(c1)CCC2)c1ccccc1

nearest known ligand 0.51

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
MLNR O43193 8/20 0.51
CYP2D6 P10635 4/20 0.44
DRD2 P14416 3/20 0.43
DRD3 P35462 3/20 0.43
TPSAB1 Q15661 1/20 0.42
ALDH1A1 P00352 1/20 0.39
HTR2C P28335 1/20 0.39
HTR2B P41595 1/20 0.39
MAPT P10636 1/20 0.39
PSIP1 O75475 1/20 0.38
HTR6 P50406 1/20 0.38
KDM4E B2RXH2 1/20 0.38
TDP1 Q9NUW8 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7854631 0.88 MLNR (0.52) MLNRCYP2D6DRD2DRD3TPSAB1
SCHEMBL7860289 0.85 MLNR (0.52) MLNRCYP2D6DRD2DRD3TPSAB1
SCHEMBL12608373 0.78 HRH3 (0.51) MLNRCYP2D6DRD2DRD3HTR2C
SCHEMBL7862464 0.77 TPSAB1 (0.47) TPSAB1ALDH1A1HTR2CHTR2BMAPT
SCHEMBL1789401 0.76 MLNR (0.74) MLNRCYP2D6HTR2CHTR2BHTR6
SCHEMBL7854715 0.75 ALDH1A1 (0.46) TPSAB1ALDH1A1HTR2CHTR2BMAPT
SCHEMBL20097742 0.74 DRD1 (0.49) MLNRCYP2D6DRD2DRD3HTR2C
SCHEMBL7861299 0.74 NPC1 (0.44) CYP2D6ALDH1A1MAPTKDM4E
SCHEMBL7862501 0.74 NPC1 (0.41) CYP2D6TPSAB1ALDH1A1HTR2CHTR2B
SCHEMBL12651580 0.74 MLNR (0.50) MLNRCYP2D6DRD2DRD3ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0807101-B1 2-AMINOINDANS AS SELECTIVE DOPAMINE D3 LIGANDS UPJOHN CO (US) 2001-06-13 EP disclosed
US-5936000-A 2-aminoindans as selective dopamine D3 ligands PHARMACIA & UPJOHN COMPANY (US) 1999-08-10 US disclosed
WO-1996023760-A1 2-AMINOINDANS AS SELECTIVE DOPAMINE D3 LIGANDS PHARMACIA & UPJOHN COMPANY (US) 1996-08-08 WO disclosed