SCHEMBL7860433

SCHEMBL7860433

CCCCc1oc2ccccc2c1C(=O)c1cc(I)c(OCCNCC(=O)O)c(I)c1

nearest known ligand 0.85

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ABCB1 P08183 2/20 0.85
SIRT3 Q9NTG7 9/20 0.79
THRA P10827 2/20 0.78
THRB P10828 2/20 0.78
KDM5A P29375 7/20 0.74
KDM4A O75164 3/20 0.74
ING2 Q9H160 1/20 0.74
KDM7A Q6ZMT4 2/20 0.70
ALDH1A1 P00352 2/20 0.70
TP53 P04637 2/20 0.70
CYP3A4 P08684 2/20 0.70
SMN1; SMN2 Q16637 2/20 0.70
TDP1 Q9NUW8 2/20 0.70
MLNR O43193 1/20 0.70
CACNA1F O60840 1/20 0.70
PHF2 O75151 1/20 0.70
ABCB11 O95342 1/20 0.70
NR3C1 P04150 1/20 0.70
ERBB2 P04626 1/20 0.70
CYP1A2 P05177 1/20 0.70

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Desethylamiodarone SCHEMBL4535165 0.92 ABCB1 (1.00) ABCB1SIRT3THRATHRBKDM5A
SCHEMBL9094309 0.92 ABCB1 (0.89) ABCB1SIRT3THRATHRBKDM5A
Desethylamiodarone SCHEMBL10673876 0.91 ABCB1 (0.95) ABCB1SIRT3THRATHRBKDM5A
Desethylamiodarone SCHEMBL10680807 0.91 ABCB1 (0.98) ABCB1SIRT3THRATHRBKDM5A
Desethylamiodarone SCHEMBL15618727 0.90 ABCB1 (0.96) ABCB1SIRT3THRATHRBKDM5A
SCHEMBL9165920 0.90 THRA (0.82) ABCB1SIRT3THRATHRBKDM5A
SCHEMBL3228984 0.88 THRA (1.00) ABCB1SIRT3THRATHRBKDM5A
SCHEMBL25873319 0.88 KDM5A (0.86) ABCB1SIRT3THRATHRBKDM5A
SCHEMBL19895690 0.87 KDM5A (0.85) ABCB1SIRT3THRATHRBKDM5A
SCHEMBL23815659 0.87 ABCB1 (0.90) ABCB1SIRT3THRATHRBKDM5A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1086063-A4 NOVEL POTASSIUM CHANNEL DRUGS AND THEIR USES ADVANCED MEDICINE INC (US) 2001-03-28 EP disclosed
EP-1086063-A1 NOVEL POTASSIUM CHANNEL DRUGS AND THEIR USES Advanced Medicine, Inc. (US) 2001-03-28 EP disclosed
WO-1999064050-A9 NOVEL POTASSIUM CHANNEL DRUGS AND THEIR USES ADVANCED MEDICINE INC (US) 2000-04-20 WO disclosed
WO-1999064050-A1 NOVEL POTASSIUM CHANNEL DRUGS AND THEIR USES ADVANCED MEDICINE, INC. (US) 1999-12-16 WO disclosed