2-Picolinic Acid

2-Picolinic Acid

SCHEMBL7860593

NC(=O)c1ccc(NC(=S)Nc2ccc(Cl)c(C(F)(F)F)c2)cc1.O=C(O)c1ccccn1

nearest known ligand 0.65

Full drug profile on Sugi Atlas →

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
GRM4 Q14833 4/20 0.65
KDR P35968 8/20 0.51
BRAF P15056 3/20 0.51
FLT3 P36888 2/20 0.51
KIT P10721 1/20 0.51
RAF1 P04049 1/20 0.51
EGFR P00533 1/20 0.49
ALDH1A1 P00352 2/20 0.49
GAA P10253 2/20 0.49
MAPT P10636 2/20 0.49
MEN1 O00255 1/20 0.49
RAB9A P51151 1/20 0.49
KMT2A Q03164 1/20 0.49
SMN1; SMN2 Q16637 1/20 0.49
HKDC1 Q2TB90 1/20 0.49
LMNA P02545 2/20 0.45
RIPK1 Q13546 1/20 0.44
TRPV1 Q8NER1 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
2-Picolinic Acid SCHEMBL7860597 0.90 GRM4 (0.67) GRM4KDRBRAFFLT3KIT
SCHEMBL7178922 0.87 GRM4 (0.86) GRM4KDRBRAFFLT3KIT
SCHEMBL6815777 0.85 KDR (0.61) GRM4KDRBRAFFLT3KIT
SCHEMBL6815026 0.77 ALDH1A1 (0.51) KDRBRAFFLT3KITALDH1A1
SCHEMBL7162138 0.76 KDR (0.78) KDRRAF1TRPV1
SCHEMBL8562560 0.76 BRAF (0.64) GRM4KDRBRAFFLT3KIT
SCHEMBL6816279 0.74 LMNA (0.60) KDRALDH1A1GAAMAPTMEN1
SCHEMBL7981202 0.74 MAPK14 (0.56) GRM4KDRALDH1A1GAAMAPT
SCHEMBL4555026 0.73 LMNA (0.75) GRM4KDRBRAFRAF1ALDH1A1
SCHEMBL7570587 0.73 BRAF (0.55) GRM4KDRBRAFALDH1A1GAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1137645-A2 ALPHA-METHYLBENZYL-CONTAINING THIOUREA INHIBITORS OF HERPES VIRUSES CONTAINING A PHENYLENEDIAMINE GROUP AMERICAN HOME PRODUCTS CORPORATION (US) 2001-10-04 EP disclosed
WO-2000034260-A2 ALPHA-METHYLBENZYL-CONTAINING THIOUREA INHIBITORS OF HERPES VIRUSES CONTAINING A PHENYLENEDIAMINE GROUP AMERICAN HOME PRODUCTS CORPORATION (US) 2000-06-15 WO disclosed