SCHEMBL7860657

SCHEMBL7860657

Cc1cc(F)cc(-c2nc(C(F)(F)F)cn2NS(=O)(=O)c2ccccc2)c1

nearest known ligand 0.54

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
PTGS2 P35354 17/20 0.54
PTGS1 P23219 7/20 0.53
SYK P43405 2/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Benzenesulfonamide SCHEMBL7050658 0.95 PTGS2 (0.62) PTGS2PTGS1
Imidazole SCHEMBL7930105 0.90 PTGS2 (0.46) PTGS2PTGS1SYK
SCHEMBL8347213 0.88 PTGS2 (0.55) PTGS2PTGS1SYK
SCHEMBL8348990 0.84 PTGS2 (0.54) PTGS2PTGS1SYK
Benzenesulfonamide SCHEMBL7932083 0.80 PTGS2 (0.62) PTGS2PTGS1
Benzenesulfonamide SCHEMBL7189185 0.79 PTGS2 (0.61) PTGS2PTGS1
SCHEMBL8025611 0.79 PTGS2 (0.55) PTGS2PTGS1
SCHEMBL7932077 0.79 PTGS2 (0.55) PTGS2PTGS1
SCHEMBL8346344 0.77 PTGS2 (0.55) PTGS2PTGS1
SCHEMBL8350247 0.77 PTGS2 (0.55) PTGS2PTGS1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1140181-A1 COMBINATION THERAPY OF RADIATION AND A COX-2 INHIBITOR FOR THE TREATMENT OF NEOPLASIA G.D. SEARLE & CO. (US) 2001-10-10 EP claimed
WO-2000038716-A1 COMBINATION THERAPY OF RADIATION AND A COX-2 INHIBITOR FOR THE TREATMENT OF NEOPLASIA G.D. SEARLE & CO. (US) 2000-07-06 WO claimed