SCHEMBL7860971

SCHEMBL7860971

N#C[CH]c1ccccc1Br

nearest known ligand 0.42

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
HSD11B1 P28845 3/20 0.42
IKBKB O14920 1/20 0.37
DYRK2 Q92630 1/20 0.37
MAPT P10636 3/20 0.36
TP53 P04637 1/20 0.36
POLB P06746 2/20 0.35
CYP1A1 P04798 2/20 0.33
CYP1A2 P05177 2/20 0.33
CYP1B1 Q16678 2/20 0.33
ALDH1A1 P00352 2/20 0.33
SMN1; SMN2 Q16637 1/20 0.33
BCHE P06276 1/20 0.33
KMT2A Q03164 3/20 0.33
ATM Q13315 1/20 0.33
LY96 Q9Y6Y9 1/20 0.33
TRPA1 O75762 1/20 0.32
MEN1 O00255 2/20 0.31
MAPK1 P28482 1/20 0.31
GAA P10253 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21457575 0.77 HSD11B1 (0.48) HSD11B1IKBKBDYRK2MAPTTP53
SCHEMBL2000509 0.77 HSD11B1 (0.48) HSD11B1IKBKBDYRK2MAPTTP53
SCHEMBL3220923 0.76 HSD11B1 (0.42) HSD11B1IKBKBDYRK2MAPTTP53
SCHEMBL5742413 0.72 HSD11B1 (0.36) HSD11B1POLBBCHE
SCHEMBL7224974 0.71 TSHR (0.50) MAPTTP53CYP1A2ALDH1A1SMN1; SMN2
SCHEMBL22440499 0.71 TRPA1 (0.32) ALDH1A1KMT2ATRPA1MEN1
SCHEMBL5415180 0.71 NFE2L2 (0.54) IKBKBDYRK2MAPK1
SCHEMBL7865931 0.71 TRPA1 (0.55) DYRK2MAPTTP53CYP1A1CYP1A2
SCHEMBL3368866 0.71 TRPA1 (0.60) HSD11B1MAPTTP53POLBCYP1A2
Acetonitrile SCHEMBL28192655 0.71 KMT2A (0.48) HSD11B1IKBKBDYRK2MAPTTP53

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1086107-A1 ARTEMISININ DERIVATIVES, METHOD FOR THE PREPARATION THEREOF AND PHARMACEUTICAL COMPOSITIONS CONTAINING THE SAME SHANGHAI INSTITUTE OF MATERIA MEDICA, CHINESE ACADEMY OF SCIENCES (CN) 2001-03-28 EP disclosed
WO-1999065914-A1 ARTEMISININ DERIVATIVES, METHOD FOR THE PREPARATION THEREOF AND PHARMACEUTICAL COMPOSITIONS CONTAINING THE SAME SHANGHAI INSTITUTE OF MATERIA MEDICA (CN) 1999-12-23 WO disclosed