SCHEMBL7861819

SCHEMBL7861819

CC(N)c1cccc([N+](=O)[O-])c1C(=O)OC(C)(C)C

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.42
TDP1 Q9NUW8 3/20 0.41
L3MBTL1 Q9Y468 1/20 0.41
NPSR1 Q6W5P4 1/20 0.38
NR3C2 P08235 1/20 0.38
HTT P42858 1/20 0.37
CYP1A2 P05177 3/20 0.37
GRM8 O00222 1/20 0.37
GRM4 Q14833 1/20 0.37
MET P08581 1/20 0.36
SLC7A5 Q01650 1/20 0.36
GPR35 Q9HC97 1/20 0.36
TSHR P16473 2/20 0.35
GLA P06280 2/20 0.35
MEN1 O00255 1/20 0.35
POLB P06746 1/20 0.35
CYP3A4 P08684 1/20 0.35
CYP2D6 P10635 1/20 0.35
MAPT P10636 1/20 0.35
CYP2C9 P11712 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17335345 0.85 ALDH1A1 (0.43) ALDH1A1TDP1L3MBTL1NPSR1NR3C2
SCHEMBL283121 0.80 ALDH1A1 (0.47) ALDH1A1TDP1L3MBTL1NPSR1NR3C2
SCHEMBL17335057 0.79 TDP1 (0.62) ALDH1A1TDP1L3MBTL1NPSR1NR3C2
SCHEMBL17827834 0.78 TDP1 (0.45) ALDH1A1TDP1L3MBTL1NPSR1NR3C2
SCHEMBL17335022 0.77 TDP1 (0.42) ALDH1A1TDP1L3MBTL1NPSR1HTT
SCHEMBL28196232 0.77 TDP1 (0.44) ALDH1A1TDP1L3MBTL1NPSR1NR3C2
SCHEMBL17334745 0.76 ERN1 (0.51) ALDH1A1TDP1L3MBTL1NPSR1HTT
SCHEMBL10402187 0.74 CTSB (0.36) ALDH1A1TDP1L3MBTL1NR3C2HTT
SCHEMBL10402188 0.74 CTSB (0.36) ALDH1A1TDP1L3MBTL1NR3C2HTT
SCHEMBL16811748 0.72 ALDH1A1 (0.56) ALDH1A1TDP1L3MBTL1NPSR1HTT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1067928-A4 METHODS FOR INHIBITING MRP1 LILLY CO ELI (US) 2001-11-14 EP disclosed
EP-1067928-A1 METHODS FOR INHIBITING MRP1 ELI LILLY AND COMPANY (US) 2001-01-17 EP disclosed
WO-1999051228-A1 METHODS FOR INHIBITING MRP1 ELI LILLY AND COMPANY (US) 1999-10-14 WO disclosed