SCHEMBL7862046

SCHEMBL7862046

N=C(N)Nc1cccc(S(=O)(=O)Nc2cccc(C(CC(=O)O)c3ccccc3)c2)c1

nearest known ligand 0.45

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
ITGB3 P05106 3/20 0.45
ITGAV P06756 3/20 0.45
MEN1 O00255 2/20 0.44
KMT2A Q03164 2/20 0.44
CA1 P00915 3/20 0.44
CA2 P00918 3/20 0.44
PKM P14618 2/20 0.43
HTR6 P50406 3/20 0.43
POLB P06746 1/20 0.42
PFKFB3 Q16875 1/20 0.42
MAPT P10636 1/20 0.42
F2 P00734 1/20 0.42
F10 P00742 1/20 0.42
PRSS1 P07477 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7864759 0.93 MEN1 (0.48) ITGB3ITGAVMEN1KMT2ACA1
SCHEMBL7856530 0.91 CA1 (0.54) ITGB3ITGAVMEN1KMT2ACA1
SCHEMBL7856528 0.91 MEN1 (0.43) ITGB3ITGAVMEN1KMT2ACA1
SCHEMBL7863164 0.91 MEN1 (0.43) ITGB3ITGAVMEN1KMT2ACA1
SCHEMBL13715863 0.90 PKM (0.46) ITGB3ITGAVMEN1KMT2ACA1
SCHEMBL7864762 0.90 CA1 (0.42) ITGB3ITGAVMEN1KMT2ACA1
SCHEMBL7864212 0.90 MEN1 (0.41) ITGB3ITGAVMEN1KMT2ACA1
SCHEMBL7863291 0.89 ITGB3 (0.45) ITGB3ITGAVMEN1KMT2ACA1
SCHEMBL7190239 0.88 ALDH1A1 (0.40) ITGB3ITGAVMEN1KMT2ACA1
SCHEMBL6366667 0.87 ITGB3 (0.60) ITGB3ITGAVCA1CA2PKM

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0889877-B1 META-SUBSTITUTED PHENYLENE DERIVATIVES AND THEIR USE AS ALPHAvBETA3 INTEGRIN ANTAGONISTS OR INHIBITORS SEARLE & CO (US) 2001-08-29 EP claimed
EP-0889877-B1 META-SUBSTITUTED PHENYLENE DERIVATIVES AND THEIR USE AS ALPHAvBETA3 INTEGRIN ANTAGONISTS OR INHIBITORS SEARLE & CO (US) 2001-08-29 EP disclosed