SCHEMBL7864175

SCHEMBL7864175

CCC(CNC(=O)c1cccc(NC(=N)N)c1)C(CC(=O)O)c1ccccc1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 1/20 0.47
LMNA P02545 2/20 0.44
ITGB3 P05106 3/20 0.43
ITGA2B P08514 2/20 0.43
F3 P13726 2/20 0.43
PKM P14618 1/20 0.42
PARP1 P09874 1/20 0.42
PARP10 Q53GL7 1/20 0.42
PAX8 Q06710 1/20 0.41
L3MBTL1 Q9Y468 1/20 0.40
MEN1 O00255 1/20 0.40
GAA P10253 1/20 0.40
KMT2A Q03164 1/20 0.40
KCNK3 O14649 1/20 0.40
KCNK9 Q9NPC2 1/20 0.40
ITGAV P06756 1/20 0.40
BCHE P06276 1/20 0.39
PLAU P00749 1/20 0.39
PRSS1 P07477 1/20 0.39
PRSS2 P07478 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7862019 0.78 LMNA (0.45) ALDH1A1LMNAITGB3ITGA2BPKM
SCHEMBL7864172 0.78 TP53 (0.46) ALDH1A1LMNAITGB3ITGA2BPARP1
SCHEMBL7856433 0.77 ITGB3 (0.54) ITGB3ITGA2BPARP1PARP10MEN1
SCHEMBL242674 0.76 ITGB3 (0.55) ITGB3ITGA2BMEN1KMT2AITGAV
SCHEMBL7863288 0.76 SIRT2 (0.48) ALDH1A1LMNAITGB3ITGA2BL3MBTL1
SCHEMBL6775429 0.76 ITGB3 (0.44) LMNAITGB3ITGA2BPARP1PARP10
SCHEMBL7455765 0.76 ITGB3 (0.58) ALDH1A1ITGB3ITGA2BMEN1KMT2A
SCHEMBL8531696 0.76 MAPT (0.48) LMNAITGB3ITGA2BPAX8KCNK3
SCHEMBL19426798 0.76 PLK4 (0.48) LMNAMEN1GAAKMT2AKCNK3
SCHEMBL7099298 0.76 ITGB3 (0.66) ITGB3ITGA2BITGAV

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0889877-B1 META-SUBSTITUTED PHENYLENE DERIVATIVES AND THEIR USE AS ALPHAvBETA3 INTEGRIN ANTAGONISTS OR INHIBITORS SEARLE & CO (US) 2001-08-29 EP claimed
EP-0889877-A1 META-SUBSTITUTED PHENYLENE DERIVATIVES AND THEIR USE AS ALPHAvBETA3 INTEGRIN ANTAGONISTS OR INHIBITORS G.D. SEARLE & CO. (US) 1999-01-13 EP claimed
WO-1997036862-A1 META-SUBSTITUTED PHENYLENE DERIVATIVES AND THEIR USE AS ALPHAvBETA3 INTEGRIN ANTAGONISTS OR INHIBITORS G.D. SEARLE & CO. (US) 1997-10-09 WO claimed
EP-0889877-B1 META-SUBSTITUTED PHENYLENE DERIVATIVES AND THEIR USE AS ALPHAvBETA3 INTEGRIN ANTAGONISTS OR INHIBITORS SEARLE & CO (US) 2001-08-29 EP disclosed