SCHEMBL7865030

SCHEMBL7865030

Cc1ncc(Cn2c(NC3CCN([C@H]4CCN[C@H](Cc5ccccc5)C4)CC3)nc3ccccc32)o1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SSTR5 P35346 7/20 0.44
KCNH2 Q12809 11/20 0.41
NR4A2 P43354 2/20 0.41
LMNA P02545 2/20 0.37
GAA P10253 2/20 0.37
MEN1 O00255 1/20 0.37
MLNR O43193 1/20 0.37
CACNA1F O60840 1/20 0.37
EED O75530 1/20 0.37
USP2 O75604 1/20 0.37
ABCB11 O95342 1/20 0.37
EGFR P00533 1/20 0.37
HLA-A P04439 1/20 0.37
ERBB2 P04626 1/20 0.37
TP53 P04637 1/20 0.37
CYP1A2 P05177 1/20 0.37
LCK P06239 1/20 0.37
FYN P06241 1/20 0.37
CHRM2 P08172 1/20 0.37
CHRM4 P08173 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7865027 1.00 SSTR5 (0.44) SSTR5KCNH2NR4A2LMNAGAA
SCHEMBL7864982 0.90 KCNH2 (0.45) SSTR5KCNH2NR4A2LMNAGAA
SCHEMBL7864978 0.90 KCNH2 (0.45) SSTR5KCNH2NR4A2LMNAGAA
SCHEMBL8162459 0.79 SSTR5 (0.48) SSTR5KCNH2NR4A2LMNAGAA
SCHEMBL9303969 0.79 KCNH2 (0.60) SSTR5KCNH2NR4A2LMNAGAA
SCHEMBL7854840 0.79 TACR1 (0.39) SSTR5LMNAGAATACR1ALDH1A1
Water SCHEMBL9302746 0.78 KCNH2 (0.48) SSTR5KCNH2NR4A2LMNAGAA
Water SCHEMBL9303352 0.78 KCNH2 (0.48) SSTR5KCNH2NR4A2LMNAGAA
Water SCHEMBL9303347 0.78 KCNH2 (0.48) SSTR5KCNH2NR4A2LMNAGAA
SCHEMBL7862726 0.78 KCNH2 (0.46) SSTR5KCNH2NR4A2LMNAGAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0869955-B1 N-ACYL-2-SUBSTITUTED-4-(BENZIMIDAZOLYL- OR IMIDAZOPYRIDINYL-SUBSTITUTED RESIDUES)-PIPERIDINES AS TACHYKININ ANTAGONISTS JANSSEN PHARMACEUTICA NV (BE) 2001-10-24 EP disclosed
US-6110939-A AS A SUBSTANCE P ANTAGONISTS TREATING TACHYKININ-MEDIATED DISEASE, ASTHMA, CENTRAL NERVOUS SYSTEM DISORDER JANSSEN PHARMACEUTICA N.V. (BE) 2000-08-29 US disclosed