Phthalic Acid

Phthalic Acid

SCHEMBL7865014

CC(C)N1CC=C(c2cc3cc([N+](=O)[O-])ccc3s2)CC1.O=C(O)c1ccccc1C(=O)O

nearest known ligand 0.44

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Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 5/20 0.44
ALDH1A1 P00352 4/20 0.44
MEN1 O00255 4/20 0.44
GAA P10253 3/20 0.44
MAPT P10636 3/20 0.44
BLM P54132 2/20 0.44
RAD52 P43351 1/20 0.44
MCL1 Q07820 1/20 0.44
SMN1; SMN2 Q16637 5/20 0.41
POLB P06746 3/20 0.41
LMNA P02545 2/20 0.41
KCNH2 Q12809 1/20 0.39
HRH3 Q9Y5N1 1/20 0.39
CYP1A2 P05177 1/20 0.37
CYP2C9 P11712 1/20 0.37
HPGD P15428 1/20 0.37
CYP2C19 P33261 1/20 0.37
AKR1B1 P15121 1/20 0.37
KDM4E B2RXH2 1/20 0.37
RAB9A P51151 3/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Phthalic Acid SCHEMBL7865021 1.00 KMT2A (0.44) KMT2AALDH1A1MEN1GAAMAPT
Fumaric Acid SCHEMBL7870869 0.81 ALDH1A1 (0.38) KMT2AALDH1A1MEN1GAAMAPT
Maleic Acid SCHEMBL7870864 0.81 ALDH1A1 (0.38) KMT2AALDH1A1MEN1GAAMAPT
Maleic Acid SCHEMBL7868007 0.72 SLC9A1 (0.38) KMT2AALDH1A1MEN1GAAMAPT
Maleic Acid SCHEMBL7865036 0.72 KDM4E (0.37) KMT2AALDH1A1MEN1GAAMAPT
Maleic Acid SCHEMBL7867476 0.70 SLC6A4 (0.41) KMT2AALDH1A1MEN1GAAMAPT
Fumaric Acid SCHEMBL7867483 0.70 SLC6A4 (0.41) KMT2AALDH1A1MEN1GAAMAPT
Fumaric Acid SCHEMBL8819859 0.70 ALDH1A1 (0.32) KMT2AALDH1A1MEN1GAAMAPT
Maleic Acid SCHEMBL8819856 0.70 ALDH1A1 (0.32) KMT2AALDH1A1MEN1GAAMAPT
Fumaric Acid SCHEMBL7865133 0.69 CYP19A1 (0.45) KMT2AALDH1A1MEN1GAAMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1077213-A2 Inhibition of serotonin reuptake ELI LILLY AND COMPANY (US) 2001-02-21 EP disclosed
US-6046215-A A PIPERIDINYLBENZOTHIOPHENES USEFUL FOR TRATING BRAIN DISORDERS ELI LILLY AND COMPANY (US) 2000-04-04 US disclosed
US-5846982-A Inhibition of serotonin reuptake ELI LILLY AND COMPANY (US) 1998-12-08 US disclosed
EP-0812826-A1 1H-indole and benzo(b)thiophene derivatives with 4-(1,2,3,6-tetra:hydro:pyridinyl)- and 4-piperidinyl-groups bound to the heterocyclic ring as inhibitors of serotonin reuptake ELI LILLY AND COMPANY (US) 1997-12-17 EP disclosed