Oxalic Acid

Oxalic Acid

SCHEMBL7865026

Clc1ccc2sc(C3=CCNCC3)cc2c1.O=C(O)C(=O)O

nearest known ligand 0.44

Full drug profile on Sugi Atlas →

Known targets — ChEMBL curated mechanism

OPRM1SLC6A4

The experimentally established mechanism targets of Oxalic Acid. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
SIGMAR1 Q99720 2/20 0.44
HTR2C P28335 5/20 0.43
HTR6 P50406 8/20 0.39
MAPT P10636 1/20 0.39
HTR1B P28222 1/20 0.39
HTR2A P28223 1/20 0.39
HTR7 P34969 1/20 0.39
HTR3A P46098 1/20 0.39
FTO Q9C0B1 1/20 0.37
MAPKAPK2 P49137 1/20 0.36
QDPR P09417 2/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7867297 0.92 SIGMAR1 (0.51) SIGMAR1HTR2CHTR6MAPTHTR1B
SCHEMBL7864911 0.82 SIGMAR1 (0.51) SIGMAR1HTR2CHTR6MAPTHTR1B
SCHEMBL5756400 0.77 HTR6 (0.44) SIGMAR1HTR2CHTR6HTR2AHTR7
Oxalic Acid SCHEMBL7859566 0.76 SLC6A4 (0.42) HTR6HTR3AQDPR
SCHEMBL4359750 0.74 SIGMAR1 (0.50) SIGMAR1HTR2CMAPTQDPR
Hydrochloric Acid SCHEMBL8321976 0.73 HTR2C (0.51) SIGMAR1HTR2CMAPTQDPR
SCHEMBL5756794 0.69 GHSR (0.33) HTR3A
SCHEMBL5758301 0.69 HTR6 (0.44) SIGMAR1HTR2CHTR6HTR2AHTR7
Hydrochloric Acid SCHEMBL8709798 0.68 DRD4 (0.53) SIGMAR1HTR2CHTR6MAPTHTR1B
SCHEMBL5760747 0.68 HTR2A (0.33) HTR2CHTR2AHTR3A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1077213-A2 Inhibition of serotonin reuptake ELI LILLY AND COMPANY (US) 2001-02-21 EP disclosed
US-6046215-A A PIPERIDINYLBENZOTHIOPHENES USEFUL FOR TRATING BRAIN DISORDERS ELI LILLY AND COMPANY (US) 2000-04-04 US disclosed
US-5846982-A Inhibition of serotonin reuptake ELI LILLY AND COMPANY (US) 1998-12-08 US disclosed
EP-0812826-A1 1H-indole and benzo(b)thiophene derivatives with 4-(1,2,3,6-tetra:hydro:pyridinyl)- and 4-piperidinyl-groups bound to the heterocyclic ring as inhibitors of serotonin reuptake ELI LILLY AND COMPANY (US) 1997-12-17 EP disclosed