SCHEMBL7866429

SCHEMBL7866429

OC1(c2cc3ccccc3[nH]2)CCN(Cc2ccccc2)CC1

nearest known ligand 0.57

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
OPRL1 P41146 3/20 0.57
POLB P06746 1/20 0.56
CCR3 P51677 1/20 0.52
KMT2A Q03164 3/20 0.52
KDM4E B2RXH2 1/20 0.52
MEN1 O00255 1/20 0.49
ALDH1A1 P00352 1/20 0.49
CYP2C9 P11712 1/20 0.49
TSHR P16473 1/20 0.49
CYP2C19 P33261 1/20 0.49
HIF1A Q16665 1/20 0.49
CYP3A4 P08684 1/20 0.46
HSD17B10 Q99714 1/20 0.46
CYP2D6 P10635 1/20 0.45
HDAC6 Q9UBN7 1/20 0.44
CHRM2 P08172 1/20 0.44
CHRM3 P20309 1/20 0.44
HRH4 Q9H3N8 1/20 0.44
SIGMAR1 Q99720 1/20 0.44
KDR P35968 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8820630 0.83 HTR6 (0.51) OPRL1POLBKMT2AMEN1ALDH1A1
SCHEMBL7500375 0.79 HRH4 (0.52) HRH4KDR
SCHEMBL12948668 0.75 FLT3 (0.41) KDM4EALDH1A1HSD17B10HRH4
SCHEMBL8681808 0.75 HRH4 (0.73) KMT2AHRH4SIGMAR1
SCHEMBL6042898 0.74 KMT2A (0.82) OPRL1POLBCCR3KMT2AKDM4E
SCHEMBL1411499 0.74 OPRL1 (1.00) OPRL1POLBCCR3KMT2AKDM4E
SCHEMBL14188677 0.73 HRH4 (0.78) POLBHDAC6HRH4SIGMAR1
Hydrochloric Acid SCHEMBL8681674 0.72 HRH4 (0.76) POLBHDAC6HRH4SIGMAR1
SCHEMBL28548988 0.71 OPRL1 (0.71) OPRL1POLBCCR3KMT2AMEN1
SCHEMBL6709096 0.71 OPRL1 (0.63) OPRL1POLBCCR3KMT2AKDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1077213-A2 Inhibition of serotonin reuptake ELI LILLY AND COMPANY (US) 2001-02-21 EP disclosed
US-6046215-A A PIPERIDINYLBENZOTHIOPHENES USEFUL FOR TRATING BRAIN DISORDERS ELI LILLY AND COMPANY (US) 2000-04-04 US disclosed
US-5846982-A Inhibition of serotonin reuptake ELI LILLY AND COMPANY (US) 1998-12-08 US disclosed
EP-0812826-A1 1H-indole and benzo(b)thiophene derivatives with 4-(1,2,3,6-tetra:hydro:pyridinyl)- and 4-piperidinyl-groups bound to the heterocyclic ring as inhibitors of serotonin reuptake ELI LILLY AND COMPANY (US) 1997-12-17 EP disclosed