SCHEMBL7867384

SCHEMBL7867384

O=S(=O)(c1ccccc1)n1c(C2=CCN(Cc3ccccc3)CC2)cc2ccccc21

nearest known ligand 0.59

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
HTR6 P50406 2/20 0.59
CA12 O43570 3/20 0.46
CA9 Q16790 3/20 0.46
CA2 P00918 1/20 0.46
DRD4 P21917 7/20 0.43
DRD3 P35462 6/20 0.43
DRD2 P14416 6/20 0.43
HTR1A P08908 1/20 0.42
HTR2A P28223 1/20 0.42
HTT P42858 1/20 0.42
ALDH1A1 P00352 2/20 0.41
PKM P14618 1/20 0.41
KDM4E B2RXH2 1/20 0.41
OPRM1 P35372 1/20 0.41
OPRK1 P41145 1/20 0.41
USP2 O75604 1/20 0.40
CYP2D6 P10635 1/20 0.40
HDAC4 P56524 1/20 0.39
NAMPT P43490 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Oxalic Acid SCHEMBL7867764 0.96 HTR6 (0.55) HTR6CA12CA9CA2DRD4
SCHEMBL7085731 0.74 HTR6 (0.53) HTR6DRD4DRD2HTR1AHTR2A
SCHEMBL7867765 0.73 HTR6 (0.57) HTR6DRD4DRD3DRD2HTR1A
SCHEMBL13197452 0.72 CA12 (0.49) HTR6CA12CA9CA2HTT
SCHEMBL7864965 0.70 OPRL1 (0.49) HTR6ALDH1A1KDM4EUSP2CYP2D6
SCHEMBL3558164 0.70 CA12 (0.78) HTR6CA12CA9CA2HTT
SCHEMBL2395932 0.70 DRD4 (0.67) DRD4DRD3DRD2HTR1AHTR2A
SCHEMBL6042349 0.69 SIGMAR1 (0.59) DRD4DRD3DRD2HTR1AHTR2A
SCHEMBL6585625 0.67 DRD4 (0.63) DRD4DRD3DRD2HTR1AHTR2A
SCHEMBL29188191 0.67 DRD4 (0.67) DRD4DRD3DRD2HTR1AHTR2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1077213-A2 Inhibition of serotonin reuptake ELI LILLY AND COMPANY (US) 2001-02-21 EP disclosed
US-6046215-A A PIPERIDINYLBENZOTHIOPHENES USEFUL FOR TRATING BRAIN DISORDERS ELI LILLY AND COMPANY (US) 2000-04-04 US disclosed
US-5846982-A Inhibition of serotonin reuptake ELI LILLY AND COMPANY (US) 1998-12-08 US disclosed
EP-0812826-A1 1H-indole and benzo(b)thiophene derivatives with 4-(1,2,3,6-tetra:hydro:pyridinyl)- and 4-piperidinyl-groups bound to the heterocyclic ring as inhibitors of serotonin reuptake ELI LILLY AND COMPANY (US) 1997-12-17 EP disclosed