SCHEMBL7869412

SCHEMBL7869412

C=C(OCC)C(=O)OCC.c1cc2cc-2c1

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
DHODH Q02127 2/20 0.48
ALDH1A1 P00352 2/20 0.47
MAPT P10636 2/20 0.47
MEN1 O00255 2/20 0.43
KMT2A Q03164 2/20 0.43
KDM4E B2RXH2 1/20 0.43
NPC1 O15118 1/20 0.43
HPGD P15428 1/20 0.43
RAB9A P51151 1/20 0.43
SMN1; SMN2 Q16637 1/20 0.43
HSD17B10 Q99714 1/20 0.43
XPO1 O14980 2/20 0.43
CA12 O43570 1/20 0.42
CA1 P00915 1/20 0.42
CA2 P00918 1/20 0.42
CA7 P43166 1/20 0.42
CA9 Q16790 1/20 0.42
CA14 Q9ULX7 1/20 0.42
GPR35 Q9HC97 1/20 0.41
CASP1 P29466 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28133466 0.84 DHODH (0.47) DHODHALDH1A1MAPTMEN1KMT2A
Ethyl Pyruvate SCHEMBL27473316 0.81 DHODH (0.50) DHODHALDH1A1MEN1KMT2ACA12
SCHEMBL9075140 0.81 DHODH (0.48) DHODHALDH1A1MAPTMEN1KMT2A
SCHEMBL94679 0.80 ALDH1A1 (0.54) ALDH1A1MAPTMEN1KMT2ASMN1; SMN2
Hydrochloric Acid SCHEMBL27667582 0.78 ALDH1A1 (0.52) ALDH1A1MAPTMEN1KMT2ASMN1; SMN2
Ethyl Acetate SCHEMBL8096818 0.77 ALDH1A1 (0.58) DHODHALDH1A1MAPTMEN1KMT2A
SCHEMBL2631517 0.76 ALDH1A1 (0.53) DHODHALDH1A1MAPTMEN1KMT2A
SCHEMBL21065601 0.76 ALDH1A1 (0.56) DHODHALDH1A1MAPT
Ethyl Propionate SCHEMBL4243851 0.76 MAPT (0.47) DHODHALDH1A1MAPTMEN1KMT2A
Acrylic Acid Ethyl Ester SCHEMBL20449045 0.75 GSTO1 (0.45) DHODHHPGDCA12CA1CA2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6306818-B1 ESTER, THIOESTER, ORGANIC CARBONATE AND/OR THIOCARBONATE DERIVATIVES; COSMETICS, DETERGENTS, FABRIC SOFTENERS, ANTIPERSPIRANTS; SUSTAINED SCENT GIVAUDAN ROURE (INTERNATIONAL) SA (CH) 2001-10-23 US claimed
EP-0816322-A1 Fragrance precursors GIVAUDAN-ROURE (INTERNATIONAL) S.A. (CH) 1998-01-07 EP claimed
US-6306818-B1 ESTER, THIOESTER, ORGANIC CARBONATE AND/OR THIOCARBONATE DERIVATIVES; COSMETICS, DETERGENTS, FABRIC SOFTENERS, ANTIPERSPIRANTS; SUSTAINED SCENT GIVAUDAN ROURE (INTERNATIONAL) SA (CH) 2001-10-23 US disclosed
EP-0816322-A1 Fragrance precursors GIVAUDAN-ROURE (INTERNATIONAL) S.A. (CH) 1998-01-07 EP disclosed