SCHEMBL7870402

SCHEMBL7870402

Cc1ccc(Cl)c(-c2noc([C@H]3CNCC[C@H]3O)c2Br)c1F

nearest known ligand 0.42

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
REN P00797 5/20 0.42
CYP3A4 P08684 4/20 0.42
KCNH2 Q12809 4/20 0.42
HTR2A P28223 1/20 0.32
HTR2C P28335 1/20 0.32
HTR2B P41595 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7874302 0.77 REN (0.52) RENCYP3A4KCNH2HTR2A
SCHEMBL556389 0.73 REN (0.80) RENCYP3A4KCNH2
SCHEMBL20951890 0.60 NR1H4 (0.46) RENCYP3A4KCNH2
SCHEMBL7871427 0.59 REN (0.56) RENCYP3A4KCNH2HTR2A
SCHEMBL4500623 0.58 SLC6A2 (0.54) KCNH2
SCHEMBL7862960 0.58 KCNH2 (0.42) RENKCNH2HTR2A
SCHEMBL4506607 0.58 SLC6A2 (0.46) RENCYP3A4KCNH2
SCHEMBL3903970 0.56 GRK2 (0.44) CYP3A4KCNH2HTR2AHTR2CHTR2B
SCHEMBL19459164 0.56 FPR1 (0.41) RENKCNH2HTR2AHTR2CHTR2B
SCHEMBL1058913 0.56 SLC6A2 (0.44)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010114978-A1 RENIN INHIBITORS MERCK SHARP & DOHME CORP. (US) 2010-10-07 WO disclosed