SCHEMBL7870518

SCHEMBL7870518

COC(=O)Oc1ccc(C(=O)NS(=O)(=O)c2ccccc2)cn1

nearest known ligand 0.64

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
P4HTM Q9NXG6 4/20 0.64
PTGS2 P35354 5/20 0.53
PTGS1 P23219 2/20 0.52
EGFR P00533 4/20 0.48
BCL2L1 Q07817 2/20 0.44
MCL1 Q07820 2/20 0.44
ALKBH2 Q6NS38 1/20 0.44
ALKBH5 Q6P6C2 1/20 0.44
FTO Q9C0B1 1/20 0.44
MEN1 O00255 1/20 0.44
LMNA P02545 1/20 0.44
KMT2A Q03164 1/20 0.44
FLT1 P17948 1/20 0.44
FLT4 P35916 1/20 0.44
KDR P35968 1/20 0.44
L3MBTL1 Q9Y468 1/20 0.44
TDP1 Q9NUW8 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9018106 0.91 MCL1 (0.59) P4HTMEGFRBCL2L1MCL1
SCHEMBL9018334 0.91 P4HTM (0.58) P4HTMPTGS2PTGS1EGFRBCL2L1
SCHEMBL9018162 0.89 SMN1; SMN2 (0.54) P4HTMMEN1LMNAKMT2ATDP1
SCHEMBL9018466 0.88 P4HTM (0.68) P4HTMPTGS2PTGS1EGFRBCL2L1
SCHEMBL9018013 0.88 P4HTM (0.58) P4HTMPTGS2PTGS1EGFRBCL2L1
SCHEMBL9017985 0.88 P4HTM (0.66) P4HTMEGFRMEN1LMNAKMT2A
SCHEMBL9018214 0.88 P4HTM (0.55) P4HTMPTGS2PTGS1EGFRBCL2L1
SCHEMBL9018232 0.86 NPC1 (0.51) P4HTMMEN1KMT2A
SCHEMBL9018024 0.86 P4HTM (0.56) P4HTMPTGS2PTGS1EGFRBCL2L1
SCHEMBL9018503 0.86 HSD17B10 (0.50) P4HTMEGFRMEN1LMNAKMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0590520-B1 Acylsulphonamido and sulphonamidopyridine-2-carboxylic acid esters, pyridine-n-oxides thereof, a process for their preparation and their use as medicaments HOECHST AG (DE) 1996-06-12 EP claimed
EP-0590520-A1 Acylsulphonamido and sulphonamidopyridine-2-carboxylic acid esters, pyridine-n-oxides thereof, a process for their preparation and their use as medicaments HOECHST AKTIENGESELLSCHAFT (DE) 1994-04-06 EP claimed
EP-0562512-B1 Sulfonamidocarbonylpyridine-2-carboxamides and their use as medicines HOECHST AG (DE) 2001-02-21 EP disclosed
EP-0590520-B1 Acylsulphonamido and sulphonamidopyridine-2-carboxylic acid esters, pyridine-n-oxides thereof, a process for their preparation and their use as medicaments HOECHST AG (DE) 1996-06-12 EP disclosed
EP-0590520-A1 Acylsulphonamido and sulphonamidopyridine-2-carboxylic acid esters, pyridine-n-oxides thereof, a process for their preparation and their use as medicaments HOECHST AKTIENGESELLSCHAFT (DE) 1994-04-06 EP disclosed
EP-0562512-A1 Sulfonamido- and sulfonamidocarbonyl-pyridine-2-carboxamides and their pyridine-N-oxides, process for their preparation and their use as medicines HOECHST AKTIENGESELLSCHAFT (DE) 1993-09-29 EP disclosed