Oxalic Acid

Oxalic Acid

SCHEMBL7870865

CCN1CCC(c2c[nH]c3cccc(C#N)c23)CC1.O=C(O)C(=O)O

nearest known ligand 0.47

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Known targets — ChEMBL curated mechanism

OPRM1SLC6A4

The experimentally established mechanism targets of Oxalic Acid. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SLC6A4 known ✓ P31645 1/20 0.47
HTR1F P30939 2/20 0.43
DRD4 P21917 1/20 0.42
CCR2 P41597 2/20 0.42
KDM4E B2RXH2 1/20 0.41
BRD4 O60885 1/20 0.41
ALDH1A1 P00352 1/20 0.41
POLB P06746 1/20 0.41
CREBBP Q92793 1/20 0.41
NOS3 P29474 1/20 0.40
NOS1 P29475 1/20 0.40
HTR2A P28223 5/20 0.40
HTR7 P34969 5/20 0.40
DRD2 P14416 3/20 0.40
KCNH2 Q12809 2/20 0.40
HDAC3 O15379 1/20 0.38
HDAC4 P56524 1/20 0.38
HDAC1 Q13547 1/20 0.38
HDAC7 Q8WUI4 1/20 0.38
HDAC2 Q92769 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Oxalic Acid SCHEMBL7867275 0.83 SLC6A4 (0.47) SLC6A4DRD4CCR2KDM4EBRD4
Oxalic Acid SCHEMBL7867934 0.79 DRD2 (0.43) SLC6A4DRD4ALDH1A1NOS3NOS1
SCHEMBL8876262 0.78 SLC6A4 (0.57) SLC6A4CCR2
Oxalic Acid SCHEMBL7867572 0.77 SLC6A4 (0.50) SLC6A4CCR2KDM4EBRD4ALDH1A1
Oxalic Acid SCHEMBL7867428 0.77 CCNT1 (0.42) DRD4KDM4EALDH1A1NOS3NOS1
SCHEMBL14163184 0.75 DRD4 (0.54) SLC6A4DRD4NOS3NOS1DRD2
Oxalic Acid SCHEMBL7866371 0.74 DRD2 (0.43) SLC6A4DRD4ALDH1A1NOS3NOS1
Oxalic Acid SCHEMBL7864882 0.74 KDM4E (0.55) SLC6A4HTR1FKDM4EPOLBHTR2A
SCHEMBL9033610 0.74 MEN1 (0.45) SLC6A4KDM4EALDH1A1POLBHTR2A
SCHEMBL8879489 0.74 HTR2C (0.54) SLC6A4NOS3NOS1HTR6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1077213-A2 Inhibition of serotonin reuptake ELI LILLY AND COMPANY (US) 2001-02-21 EP disclosed
US-6046215-A A PIPERIDINYLBENZOTHIOPHENES USEFUL FOR TRATING BRAIN DISORDERS ELI LILLY AND COMPANY (US) 2000-04-04 US disclosed
US-5846982-A Inhibition of serotonin reuptake ELI LILLY AND COMPANY (US) 1998-12-08 US disclosed
EP-0812826-A1 1H-indole and benzo(b)thiophene derivatives with 4-(1,2,3,6-tetra:hydro:pyridinyl)- and 4-piperidinyl-groups bound to the heterocyclic ring as inhibitors of serotonin reuptake ELI LILLY AND COMPANY (US) 1997-12-17 EP disclosed