SCHEMBL7871376

SCHEMBL7871376

CCCCCC1C(C(=O)OCC#Cc2cccnc2)=C(C)NC(c2ccc(-n3c(C)nc4cnccc43)cc2)=C1C(=O)OCC

nearest known ligand 0.43

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
ADORA3 P0DMS8 3/20 0.37
TRPV1 Q8NER1 1/20 0.36
MAPT P10636 2/20 0.36
MAPK1 P28482 1/20 0.36
TSHR P16473 1/20 0.35
TMIGD3 P0DMS9 1/20 0.35
MEN1 O00255 1/20 0.35
KMT2A Q03164 1/20 0.35
NPSR1 Q6W5P4 1/20 0.35
GRM5 P41594 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7869551 0.92 ADORA3 (0.39) ADORA3TRPV1MAPTMAPK1TSHR
SCHEMBL8143535 0.92 ADORA3 (0.40) ADORA3TRPV1MAPTMAPK1TSHR
SCHEMBL7864174 0.91 ADORA3 (0.37) ADORA3TRPV1MAPTMAPK1TSHR
SCHEMBL7864163 0.91 ADORA3 (0.34) ADORA3MAPTMAPK1TSHR
SCHEMBL7873283 0.91 ADORA3 (0.40) ADORA3TRPV1MAPK1TSHRTMIGD3
SCHEMBL7872515 0.91 ADORA3 (0.38) ADORA3MAPTMAPK1TSHRTMIGD3
SCHEMBL7873250 0.90 ADORA3 (0.37) ADORA3TRPV1MAPTMAPK1TSHR
SCHEMBL7873331 0.90 MAPT (0.36) ADORA3TRPV1MAPTMAPK1TSHR
SCHEMBL7871436 0.90 TSHR (0.38) ADORA3TSHRTMIGD3GRM5
SCHEMBL7864225 0.89 ADORA3 (0.41) ADORA3MAPK1TSHRTMIGD3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6306853-B1 DICARBOXYLIC ESTER DERIVATIVES OF DIHYDROPYRIDINE COMPOUNDS NIKKEN CHEMICALS CO., LTD. (JP) 2001-10-23 US disclosed
EP-1055672-A1 1,4-DIHYDROPYRIDINE DERIVATIVES Nikken Chemicals Company, Limited (JP) 2000-11-29 EP disclosed