SCHEMBL7864174

SCHEMBL7864174

CCOC(=O)C1=C(c2ccc(-n3c(C)nc4cnccc43)cc2)NC(C)=C(C(=O)OCC#Cc2cccnc2)C1CCSC

nearest known ligand 0.42

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
ADORA3 P0DMS8 3/20 0.37
TRPV1 Q8NER1 1/20 0.36
TSHR P16473 1/20 0.35
ALDH1A1 P00352 1/20 0.35
TMIGD3 P0DMS9 1/20 0.35
GAA P10253 1/20 0.35
MAPT P10636 1/20 0.34
MAPK1 P28482 1/20 0.34
GRM5 P41594 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7871376 0.91 ADORA3 (0.37) ADORA3TRPV1TSHRTMIGD3MAPT
SCHEMBL7873283 0.90 ADORA3 (0.40) ADORA3TRPV1TSHRTMIGD3GAA
SCHEMBL7872515 0.90 ADORA3 (0.38) ADORA3TSHRTMIGD3MAPTMAPK1
SCHEMBL8143535 0.89 ADORA3 (0.40) ADORA3TRPV1TSHRTMIGD3GAA
SCHEMBL7871436 0.89 TSHR (0.38) ADORA3TSHRTMIGD3GRM5
SCHEMBL7864225 0.89 ADORA3 (0.41) ADORA3TSHRTMIGD3MAPK1
SCHEMBL7869561 0.89 ADORA3 (0.36) ADORA3TRPV1TSHRTMIGD3MAPT
SCHEMBL7869567 0.88 ALDH1A1 (0.37) ADORA3TRPV1TSHRALDH1A1TMIGD3
SCHEMBL7864163 0.88 ADORA3 (0.34) ADORA3TSHRMAPTMAPK1
SCHEMBL7869551 0.88 ADORA3 (0.39) ADORA3TRPV1TSHRTMIGD3GAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6306853-B1 DICARBOXYLIC ESTER DERIVATIVES OF DIHYDROPYRIDINE COMPOUNDS NIKKEN CHEMICALS CO., LTD. (JP) 2001-10-23 US disclosed
EP-1055672-A1 1,4-DIHYDROPYRIDINE DERIVATIVES Nikken Chemicals Company, Limited (JP) 2000-11-29 EP disclosed