SCHEMBL7871920

SCHEMBL7871920

COc1ccc(CC(N)C(O)C(=O)O)cc1

nearest known ligand 0.65

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
LDHA P00338 1/20 0.65
LTA4H P09960 2/20 0.56
SLC6A4 P31645 1/20 0.54
CYP1A2 P05177 1/20 0.51
CYP2D6 P10635 1/20 0.51
CYP2C19 P33261 1/20 0.51
PPARG P37231 1/20 0.51
PPARA Q07869 1/20 0.51
LAP3 P28838 1/20 0.51
POLB P06746 1/20 0.49
TPH1 P17752 2/20 0.48
KMT2A Q03164 1/20 0.47
CA2 P00918 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7426450 1.00 LDHA (0.65) LDHALTA4HSLC6A4CYP1A2CYP2D6
SCHEMBL20027598 0.87 LDHA (0.56) LDHALTA4HSLC6A4CYP1A2CYP2D6
SCHEMBL7961571 0.86 LTA4H (0.69) LDHALTA4HSLC6A4CYP1A2CYP2D6
SCHEMBL12379291 0.83 LTA4H (0.57) LTA4HPPARGPPARALAP3
SCHEMBL5812622 0.81 PPARG (0.48) LTA4HPPARGPPARALAP3KMT2A
SCHEMBL158667 0.81 LDHA (0.71) LDHASLC6A4CYP1A2CYP2D6CYP2C19
SCHEMBL126195 0.81 LDHA (0.71) LDHASLC6A4CYP1A2CYP2D6CYP2C19
SCHEMBL597743 0.81 LDHA (0.71) LDHASLC6A4CYP1A2CYP2D6CYP2C19
SCHEMBL7432229 0.81 LDHA (0.54) LDHALTA4HSLC6A4LAP3
SCHEMBL7432217 0.81 LDHA (0.54) LDHALTA4HSLC6A4LAP3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-1774635-A Anti-epileptogenic agents UNIV KINGSTON (CA) 2006-05-17 CN disclosed
US-6329502-B1 VIRICIDES AGAINST HUMAN IMMUNODEFICIENCY VIRUS; TREATMENT OF AIDS (ACQUIRED IMMUNE DEFICIENCY SYNDROME) JAPAN ENERGY CORPORATION (JP) 2001-12-11 US disclosed
US-6313094-B1 COMPOSITION FOR INHIBITING HUMAN IMMUNODEFICIENCY VIRUS REPLICATION JAPAN ENERGY CORPORATION (JP) 2001-11-06 US disclosed
EP-0490667-B1 HIV protease inhibitors JAPAN ENERGY CORP (JP) 1999-06-09 EP disclosed
EP-0490667-A2 HIV protease inhibitors JAPAN ENERGY CORPORATION (JP) 1992-06-17 EP disclosed