SCHEMBL7872437

SCHEMBL7872437

COc1cccc(COc2ccccc2C(C#N)NC(=O)CCC(=O)O)c1

nearest known ligand 0.54

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
SGMS2 Q8NHU3 12/20 0.54
ALDH1A1 P00352 4/20 0.54
LMNA P02545 3/20 0.54
GAA P10253 2/20 0.54
KDM4E B2RXH2 1/20 0.51
CYP1A2 P05177 1/20 0.46
CYP2C9 P11712 1/20 0.46
CYP2C19 P33261 1/20 0.46
MME P08473 1/20 0.44
SLC1A5 Q15758 1/20 0.44
ABCB1 P08183 1/20 0.43
HTR1A P08908 1/20 0.43
DRD2 P14416 1/20 0.43
FFAR1 O14842 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7872435 0.77 F2 (0.47) SGMS2ALDH1A1GAAKDM4E
SCHEMBL7872355 0.77 ABCB1 (0.54) SGMS2ALDH1A1LMNAGAAKDM4E
SCHEMBL7868630 0.69 CNR2 (0.46) GAACYP1A2CYP2C19MME
SCHEMBL7865908 0.69 HTT (0.43) CYP1A2CYP2C19MME
SCHEMBL7865923 0.69 MME (0.44) SGMS2ALDH1A1GAAKDM4ECYP1A2
SCHEMBL1388008 0.69 MRGPRX4 (0.59) ALDH1A1GAAKDM4ESLC1A5ABCB1
SCHEMBL22351829 0.67 CYP2D6 (0.65) SLC1A5ABCB1HTR1ADRD2FFAR1
SCHEMBL22351827 0.67 CYP2D6 (0.65) SLC1A5ABCB1HTR1ADRD2FFAR1
SCHEMBL21793250 0.67 CYP2D6 (0.48) SLC1A5ABCB1HTR1ADRD2FFAR1
SCHEMBL7867488 0.67 MME (0.43) ALDH1A1CYP1A2CYP2C19MME

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1086107-A1 ARTEMISININ DERIVATIVES, METHOD FOR THE PREPARATION THEREOF AND PHARMACEUTICAL COMPOSITIONS CONTAINING THE SAME SHANGHAI INSTITUTE OF MATERIA MEDICA, CHINESE ACADEMY OF SCIENCES (CN) 2001-03-28 EP disclosed
WO-1999065914-A1 ARTEMISININ DERIVATIVES, METHOD FOR THE PREPARATION THEREOF AND PHARMACEUTICAL COMPOSITIONS CONTAINING THE SAME SHANGHAI INSTITUTE OF MATERIA MEDICA (CN) 1999-12-23 WO disclosed