SCHEMBL7874467

SCHEMBL7874467

CCCc1ccc(-n2nc(Cl)cc2-c2ccc(S(C)(=O)=O)cc2)cc1[N+](=O)[O-]

nearest known ligand 0.47

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
ALOX5 P09917 2/20 0.47
PTGS2 P35354 15/20 0.44
PTGS1 P23219 2/20 0.44
CYP2C9 P11712 1/20 0.44
AOC3 Q16853 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7874491 0.94 PTGS2 (0.46) ALOX5PTGS2PTGS1CYP2C9
SCHEMBL7878975 0.88 ALOX5 (0.51) ALOX5PTGS2PTGS1CYP2C9AOC3
SCHEMBL7867762 0.85 PTGS2 (0.48) ALOX5PTGS2PTGS1CYP2C9AOC3
SCHEMBL8073636 0.83 IDO1 (0.40) ALOX5PTGS2PTGS1
SCHEMBL7876239 0.82 PTGS2 (0.48) ALOX5PTGS2PTGS1CYP2C9
SCHEMBL7878920 0.82 PTGS2 (0.56) ALOX5PTGS2PTGS1CYP2C9AOC3
SCHEMBL7876672 0.82 PTGS2 (0.50) ALOX5PTGS2PTGS1CYP2C9AOC3
SCHEMBL7879006 0.81 PTGS2 (0.52) ALOX5PTGS2PTGS1CYP2C9
SCHEMBL7876226 0.80 PTGS2 (0.48) ALOX5PTGS2PTGS1CYP2C9
SCHEMBL27556627 0.80 PTGS2 (0.57) ALOX5PTGS2PTGS1CYP2C9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6316485-B1 INHIBITS ACTIVITY OF CYCLOOXYGENASE-2; FOR THERAPY AND PROPHYLAXIS OF INFLAMMATION, THROMBOSIS, RHEUMATOID ARTHRITIS, ALZHEIMER'S DISEASE; AS ANALGESIC FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 2001-11-13 US disclosed
CN-1271347-A 1, 5-diphenylpyrazole derivatives FUJISAWA PHARMACEUTICAL CO (JP) 2000-10-25 CN disclosed