SCHEMBL78755

SCHEMBL78755

Cc1cc(N2CCOCC2)ccc1N

nearest known ligand 0.67

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
LGMN Q99538 4/20 0.67
GAA P10253 4/20 0.61
RAD52 P43351 1/20 0.61
MAPT P10636 10/20 0.58
ALDH1A1 P00352 4/20 0.58
KDM4E B2RXH2 4/20 0.58
ALOX15 P16050 3/20 0.58
TP53 P04637 3/20 0.58
MEN1 O00255 3/20 0.58
KMT2A Q03164 3/20 0.58
HTT P42858 3/20 0.58
MAPK1 P28482 3/20 0.58
HSD17B10 Q99714 2/20 0.58
USP2 O75604 1/20 0.58
SMN1; SMN2 Q16637 4/20 0.50
HPGD P15428 2/20 0.50
MITF O75030 1/20 0.50
NTSR1 P30989 1/20 0.50
NPC1 O15118 3/20 0.48
RAB9A P51151 3/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL2951905 0.98 LGMN (0.65) LGMNGAARAD52MAPTALDH1A1
SCHEMBL15358759 0.87 GAA (0.77) LGMNGAARAD52MAPTALDH1A1
SCHEMBL6151434 0.87 GAA (0.77) LGMNGAARAD52MAPTALDH1A1
SCHEMBL30545196 0.86 LGMN (0.62) LGMNGAARAD52MAPTALDH1A1
SCHEMBL375628 0.86 LGMN (0.62) LGMNGAARAD52MAPTALDH1A1
SCHEMBL19648924 0.84 LGMN (0.53) LGMNGAARAD52MAPTALDH1A1
SCHEMBL904452 0.83 LGMN (0.73) LGMNGAAMAPTALDH1A1KDM4E
SCHEMBL7032717 0.83 GAA (0.67) LGMNGAARAD52MAPTALDH1A1
SCHEMBL2923577 0.83 GAA (0.67) LGMNGAARAD52MAPTALDH1A1
SCHEMBL1911932 0.83 MAPT (0.69) LGMNGAAMAPTALDH1A1KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 211 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2050749-B1 PYRIMIDINE DERIVATIVE AS PI3K INHIBITOR AND USE THEREOF CHUGAI PHARMACEUTICAL CO LTD (JP) 2017-11-22 EP claimed
US-20100069629-A1 PYRIMIDINE DERIVATIVES AS PI3K INHIBITOR AND USE THEREOF CHUGAI SEIYAKU KABUSHIKI KAISHA (JP) 2010-03-18 US claimed
EP-2050749-A1 PYRIMIDINE DERIVATIVE AS PI3K INHIBITOR AND USE THEREOF CHUGAI SEIYAKU KABUSHIKI KAISHA (JP) 2009-04-22 EP claimed
US-20250263404-A1 AMINOPYRIDINES AS ACTIVATORS OF PI3 KINASE UCL BUSINESS LTD (GB) 2025-08-21 US disclosed
US-RE50082-E1 (5,6-dihydro)pyrimido[4,5-e]indolizines NETHERLANDS TRANSLATIONAL RESEARCH CENTER B.V. (NL) 2024-08-20 US disclosed
EP-4402127-A1 AMINOPYRIDINES AS ACTIVATORS OF PI3 KINASE UCL Business Ltd (GB) 2024-07-24 EP disclosed
US-20230365559-A1 NOVEL AMINOPYRIDINES AND THEIR USE IN TREATING CANCER AUCKLAND UNISERVICES LIMITED (NZ) 2023-11-16 US disclosed
EP-3966207-B1 PHENYLAMINOPYRIMIDINE AMIDE AUTOPHAGY INHIBITORS AND METHODS OF USE THEREOF DECIPHERA PHARMACEUTICALS LLC (US) 2023-11-01 EP disclosed
EP-4217357-A1 NOVEL AMINOPYRIDINES AND THEIR USE IN TREATING CANCER Auckland Uniservices Limited (NZ) 2023-08-02 EP disclosed
WO-2023041905-A1 AMINOPYRIDINES AS ACTIVATORS OF PI3 KINASE UCL BUSINESS LTD (GB) 2023-03-23 WO disclosed
CN-111217816-B FLT3 kinase inhibitor and preparation and application thereof 中国科学院上海药物研究所 2022-08-16 CN disclosed
EP-0181728-A2 Light-sensitive silver halide photographic material KONICA CORPORATION (JP) 1986-05-21 EP disclosed
US-4581327-A CORE AND SHELL STRUCTURES, RHODIUM DOPED SHELLS, HARDNESS OF TONE, STORAGE STABILITY KONISHIROKU PHOTO INDUSTRY CO., LTD. (JP) 1986-04-08 US disclosed
EP-0146302-A1 Light-sensitive silver halide photographic material for direct-post and method for processing the same KONICA CORPORATION (JP) 1985-06-26 EP disclosed
US-4444875-A LAYER OF A TETRAZOLIUM COMPOUND KONISHIROKU PHOTO INDUSTRY CO., LTD. (JP) 1984-04-24 US disclosed
US-4329417-A OXIDIZERS AND QUATERNARY AMMONIUM SALTS, PHOSPHONIUM SALTS OR SULFONIUM SALTS KONISHIROKU PHOTO INDUSTRY CO., LTD. (JP) 1982-05-11 US disclosed
US-4233399-A Photographic elements containing amino-substituted hydroxy-pyridones CIBA-GEIGY AKTIENGESELLSCHAFT (CH) 1980-11-11 US disclosed
US-4211835-A TETRAZOLIUM COMPOUND, BLACK AND WHITE, HIGH CONTRAST KONISHIROKU PHOTO INDUSTRY CO., LTD. (JP) 1980-07-08 US disclosed
US-4192682-A NON-DIFFUSIBLE COMPOUND HAVING OXIDATION POWER ON A HYDROQUINONE DEVELOPING AGENT; DEVELOPER CONTAINING NO HYDROQUINONE KONISHIROKU PHOTO INDUSTRY CO., LTD. (JP) 1980-03-11 US disclosed
US-4182886-A OPTICAL FILTERS IN COLOR PHOTOGRAPHY CIBA-GEIGY AKTIENGESELLSCHAFT (CH) 1980-01-08 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (3 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20100069629-A1 PYRIMIDINE DERIVATIVES AS PI3K INHIBITOR AND USE THEREOF PIK3CA, AKT3, AKT1 LGMN 4876/4885GAA 2827/4885RAD52 2095/4885
US-20230365559-A1 NOVEL AMINOPYRIDINES AND THEIR USE IN TREATING CANCER DCK, DTYMK, TYMP LGMN 4515/4885GAA 2100/4885RAD52 791/4885
US-20250263404-A1 AMINOPYRIDINES AS ACTIVATORS OF PI3 KINASE PIK3CD, PTEN, PIK3CG LGMN 4181/4885GAA 882/4885RAD52 4631/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.