SCHEMBL7876069

SCHEMBL7876069

COC(=O)C1=C(c2ccc(-n3ccnc3)cc2)NC(C)=C(C(=O)OCC#Cc2cccnc2)C1CCc1ccccc1

nearest known ligand 0.39

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
ADORA3 P0DMS8 9/20 0.39
HTT P42858 1/20 0.35
CYP3A4 P08684 3/20 0.35
CYP2D6 P10635 2/20 0.35
CYP2C9 P11712 1/20 0.35
WNT3A P56704 1/20 0.35
PORCN Q9H237 1/20 0.35
TMIGD3 P0DMS9 1/20 0.35
TRPV1 Q8NER1 2/20 0.34
ALDH1A1 P00352 2/20 0.34
NPSR1 Q6W5P4 1/20 0.34
HSD17B10 Q99714 1/20 0.34
LMNA P02545 1/20 0.34
POLB P06746 1/20 0.34
MAPK1 P28482 1/20 0.34
KMT2A Q03164 1/20 0.34
ADH5 P11766 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7871558 0.96 ADORA3 (0.43) ADORA3CYP3A4TMIGD3TRPV1ALDH1A1
SCHEMBL7872517 0.93 ADORA3 (0.38) ADORA3CYP3A4TMIGD3TRPV1ALDH1A1
SCHEMBL7871519 0.89 ADORA3 (0.37) ADORA3HTTCYP3A4CYP2D6CYP2C9
SCHEMBL7869546 0.89 ADORA3 (0.41) ADORA3HTTCYP3A4TMIGD3TRPV1
SCHEMBL7873247 0.86 ADORA3 (0.41) ADORA3CYP3A4TMIGD3TRPV1ALDH1A1
SCHEMBL7869557 0.85 ADORA3 (0.42) ADORA3CYP3A4CYP2D6CYP2C9TMIGD3
SCHEMBL7871453 0.83 ADORA3 (0.41) ADORA3CYP3A4TMIGD3TRPV1ALDH1A1
SCHEMBL7876025 0.83 ALDH1A1 (0.42) ADORA3CYP3A4TMIGD3TRPV1ALDH1A1
SCHEMBL7876057 0.83 ADORA3 (0.42) ADORA3CYP3A4TMIGD3TRPV1ALDH1A1
SCHEMBL7864230 0.82 ADORA3 (0.41) ADORA3CYP3A4CYP2C9TMIGD3TRPV1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6306853-B1 DICARBOXYLIC ESTER DERIVATIVES OF DIHYDROPYRIDINE COMPOUNDS NIKKEN CHEMICALS CO., LTD. (JP) 2001-10-23 US disclosed
EP-1055672-A1 1,4-DIHYDROPYRIDINE DERIVATIVES Nikken Chemicals Company, Limited (JP) 2000-11-29 EP disclosed